SCHEMBL9375004

SCHEMBL9375004

C=CC(O)(c1ccccc1)c1ccnn1C

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.37
KMT2A Q03164 3/20 0.36
HSP90AA1 P07900 1/20 0.35
MEN1 O00255 1/20 0.34
GPR52 Q9Y2T5 1/20 0.33
CHRM3 P20309 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.32
ACSS2 Q9NR19 1/20 0.32
NPC1 O15118 1/20 0.32
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
RAB9A P51151 1/20 0.32
ATM Q13315 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
COMT P21964 1/20 0.30
CYP3A4 P08684 1/20 0.30
MAPK1 P28482 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4910358 0.80 KDM4E (0.35) KDM4EKMT2AMEN1SMN1; SMN2ALDH1A1
SCHEMBL7752685 0.74 ALDH1A1 (0.40) KDM4EKMT2AMEN1GPR52CHRM3
SCHEMBL4887210 0.73 KDM4E (0.48) KDM4EHSP90AA1ALDH1A1CYP3A4MAPK1
SCHEMBL7755239 0.72 CHRM3 (0.38) KMT2AMEN1GPR52CHRM3ALDH1A1
SCHEMBL4902287 0.71 CYP19A1 (0.46) KMT2AACSS2L3MBTL1CYP3A4
SCHEMBL19857578 0.68 COMT (0.35) KMT2ASMN1; SMN2NPC1ALDH1A1RAB9A
SCHEMBL29140377 0.67 KDM4E (0.44) KDM4EKMT2AMEN1SMN1; SMN2ALDH1A1
SCHEMBL4909153 0.67 CNR1 (0.38) KMT2AMEN1SMN1; SMN2ALDH1A1L3MBTL1
SCHEMBL10630760 0.67 KCNA5 (0.51) KMT2AMEN1CYP3A4
SCHEMBL28395509 0.67 L3MBTL1 (0.52) KDM4EKMT2AMEN1CHRM3SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0289380-B1 Aryl-heteroaryl-carbinol derivatives having an analgesic activity ESTEVE LABOR DR (ES) 1994-12-28 EP claimed
US-5017596-A Arylpyrazolylcarbinol compounds with analgesic activity LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 1991-05-21 US claimed