SCHEMBL9375293

SCHEMBL9375293

CCC1(c2ccccc2)c2ccccc2CCN1Cc1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 15/20 0.46
TP53 P04637 2/20 0.46
CYP1A2 P05177 2/20 0.46
CYP3A4 P08684 2/20 0.46
CYP2D6 P10635 2/20 0.46
TSHR P16473 2/20 0.46
CYP2C19 P33261 2/20 0.46
DRD2 P14416 1/20 0.46
NFKB1 P19838 1/20 0.46
HTR2A P28223 1/20 0.46
HTR2C P28335 1/20 0.46
MAPK1 P28482 1/20 0.46
HTR2B P41595 1/20 0.46
MTOR P42345 1/20 0.46
MEN1 O00255 1/20 0.45
BLM P54132 1/20 0.45
PMP22 Q01453 1/20 0.45
KMT2A Q03164 1/20 0.45
ALDH1A1 P00352 1/20 0.45
CYP2C9 P11712 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2792683 0.81 SIGMAR1 (0.51) SIGMAR1TP53CYP1A2CYP3A4CYP2D6
SCHEMBL9374898 0.80 SIGMAR1 (0.48) SIGMAR1TP53CYP1A2CYP3A4CYP2D6
SCHEMBL27345750 0.77 SIGMAR1 (0.48) SIGMAR1TP53CYP1A2CYP3A4CYP2D6
SCHEMBL8840218 0.75 SIGMAR1 (0.48) SIGMAR1TP53CYP1A2CYP3A4CYP2D6
SCHEMBL1404036 0.75 MITF (0.39) MEN1KMT2A
SCHEMBL6073260 0.75 MITF (0.39) MEN1KMT2A
SCHEMBL9375323 0.74 SIGMAR1 (0.46) SIGMAR1TP53CYP1A2CYP3A4CYP2D6
SCHEMBL9374100 0.73 SIGMAR1 (0.50) SIGMAR1TP53CYP1A2CYP3A4CYP2D6
SCHEMBL9379947 0.73 SIGMAR1 (0.47) SIGMAR1TP53CYP1A2CYP3A4CYP2D6
SCHEMBL9378962 0.73 SIGMAR1 (0.49) SIGMAR1TP53CYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0336228-B1 Tetrahydroisoquinolines and tetrahydrobenzazepines and a process for the preparation thereof FUJISAWA PHARMACEUTICAL CO (JP) 1994-11-09 EP disclosed
US-5059608-A Anticonvulsants, antiischemic agents FUJISAWA PHARMACEUTICAL COMPANY, LTD. (JP) 1991-10-22 US disclosed
EP-0336228-A1 Tetrahydroisoquinolines and tetrahydrobenzazepines and a process for the preparation thereof FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1989-10-11 EP disclosed