SCHEMBL9375609

SCHEMBL9375609

Cc1ccc2c(c1)OCC(=O)N(CCCCN1CCN(c3ccccn3)CC1)C2=O

nearest known ligand 0.61

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.54
DRD2 P14416 5/20 0.54
HTR1A P08908 5/20 0.54
HTR2A P28223 4/20 0.54
HTR7 P34969 4/20 0.54
HTR6 P50406 2/20 0.54
GRIN1 Q05586 1/20 0.54
GRIN2B Q13224 1/20 0.54
DRD3 P35462 5/20 0.52
DRD1 P21728 3/20 0.52
DRD4 P21917 2/20 0.49
HTR2C P28335 2/20 0.49
SLC6A4 P31645 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9369647 0.99 KCNH2 (0.56) KCNH2DRD2HTR1AHTR2AHTR7
SCHEMBL9371971 0.90 HTR1A (0.58) DRD2HTR1AHTR2AHTR7HTR6
SCHEMBL9371995 0.90 HTR1A (0.57) DRD2HTR1AHTR2AHTR7HTR6
SCHEMBL9369094 0.89 HTR1A (0.59) DRD2HTR1AHTR2AHTR7HTR6
SCHEMBL9371917 0.88 HTR1A (0.55) DRD2HTR1AHTR2AHTR7HTR6
SCHEMBL9371795 0.87 DRD2 (0.64) KCNH2DRD2HTR1AHTR2AHTR7
SCHEMBL9372762 0.86 DRD3 (0.61) DRD2HTR1AHTR2AHTR7HTR6
SCHEMBL9369887 0.85 DRD2 (0.45) DRD2HTR1AHTR2A
SCHEMBL9373729 0.85 DRD2 (0.44) DRD2HTR1AHTR2A
SCHEMBL9369082 0.83 DRD2 (0.49) DRD2HTR1AHTR2AHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0376633-B1 Benzoxazepine derivatives SUNTORY LTD (JP) 1994-10-12 EP disclosed
US-5071845-A Psychotropic or anxyiolytic agent SUNTORY LIMITED (JP) 1991-12-10 US disclosed
EP-0376633-A2 Benzoxazepine derivatives SUNTORY LIMITED (JP) 1990-07-04 EP disclosed