SCHEMBL9375731

SCHEMBL9375731

Cc1ccc(S(=O)(=O)OCC2Cc3cccc(C)c3O2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.39
CYP2D6 P10635 3/20 0.39
CYP3A4 P08684 2/20 0.39
TSHR P16473 2/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
MAPT P10636 1/20 0.39
MAPK1 P28482 1/20 0.39
PRMT5 O14744 1/20 0.38
WDR77 Q9BQA1 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.37
CA2 P00918 1/20 0.37
PSEN1 P49768 2/20 0.35
PSEN2 P49810 2/20 0.35
APH1B Q8WW43 2/20 0.35
NCSTN Q92542 2/20 0.35
APH1A Q96BI3 2/20 0.35
PSENEN Q9NZ42 2/20 0.35
LMNA P02545 2/20 0.35
BRD4 O60885 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4227006 0.90 CA2 (0.38) ALDH1A1CYP2D6CYP3A4TSHRCYP2C9
SCHEMBL9373240 0.90 ALDH1A1 (0.38) ALDH1A1CYP2D6CYP3A4TSHRCYP2C9
SCHEMBL4220854 0.89 ALDH1A1 (0.39) ALDH1A1CYP2D6CYP3A4TSHRCYP2C9
SCHEMBL4226990 0.89 ALDH1A1 (0.41) ALDH1A1CYP2D6CYP3A4TSHRCYP2C9
SCHEMBL4225370 0.89 PRKAB2 (0.42) ALDH1A1CYP2D6CYP3A4TSHRCYP2C9
SCHEMBL4224280 0.89 ALDH1A1 (0.41) ALDH1A1CYP2D6CYP3A4TSHRCYP2C9
SCHEMBL4218710 0.89 MEN1 (0.41) ALDH1A1CYP2D6CYP3A4TSHRCYP2C9
SCHEMBL9446303 0.89 ALDH1A1 (0.39) ALDH1A1CYP2D6CYP3A4TSHRCYP2C9
SCHEMBL4226042 0.88 ALDH1A1 (0.38) ALDH1A1CYP2D6CYP3A4TSHRCYP2C9
SCHEMBL4231318 0.88 KMT2A (0.40) ALDH1A1CYP2D6CYP3A4TSHRCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0445026-B1 Aminomethylpiperidine derivatives, their process for preparation and the pharmaceutical compositions containing them ADIR (FR) 1994-01-26 EP disclosed
US-5229399-A Analgesics ADIR ET COMPAGNIE (FR) 1993-07-20 US disclosed
US-5229398-A Analgesics ADIR ET COMPAGNIE (FR) 1993-07-20 US disclosed
US-5192775-A Analgesics ADIR ET COMPAGNIE (FR) 1993-03-09 US disclosed
EP-0445026-A1 Aminomethylpiperidine derivatives, their process for preparation and the pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1991-09-04 EP disclosed