SCHEMBL9376016

SCHEMBL9376016

CC1(C)N=C(n2ccccc2=O)c2cc(N)ccc2O1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 1/20 0.34
SMN1; SMN2 Q16637 3/20 0.33
NPC1 O15118 2/20 0.32
ALDH1A1 P00352 2/20 0.32
RAB9A P51151 2/20 0.32
TP53 P04637 1/20 0.32
CYP3A4 P08684 1/20 0.32
TSHR P16473 1/20 0.32
MAPK1 P28482 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
BRPF1 P55201 1/20 0.31
PTPRC P08575 2/20 0.31
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
APAF1 O14727 1/20 0.31
TDP2 O95551 1/20 0.31
NSD2 O96028 1/20 0.31
LMNA P02545 1/20 0.31
PLA2G1B P04054 1/20 0.31
POLB P06746 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10435504 0.86 KDM4E (0.36) HRH4ALDH1A1HPGDHTTBLM
SCHEMBL9372171 0.85 F10 (0.35) HRH4SMN1; SMN2ALDH1A1TP53CYP3A4
SCHEMBL9372466 0.85 HSD11B1 (0.33) ALDH1A1CYP3A4TDP1HPGD
SCHEMBL10435505 0.85
SCHEMBL9372070 0.85 BACE1 (0.33) RAB9APTPRCMEN1KMT2AHTT
SCHEMBL9372567 0.84 ADK (0.32) HRH4ALDH1A1MEN1KMT2AHPGD
SCHEMBL9375674 0.84 F10 (0.39) SMN1; SMN2ALDH1A1TSHRBRPF1BRD4
SCHEMBL9376497 0.83 PPIB (0.44) SMN1; SMN2NPC1ALDH1A1RAB9ATP53
SCHEMBL9377805 0.83 RXFP1 (0.31) ALDH1A1
SCHEMBL9373865 0.83 F10 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0371312-B1 Benzoxazine derivatives MERCK PATENT GMBH (DE) 1994-07-20 EP disclosed
US-5036068-A Cardiovascular disorders MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1991-07-30 US disclosed
EP-0371312-A1 Benzoxazine derivatives MERCK PATENT GmbH (DE) 1990-06-06 EP disclosed