SCHEMBL9378264

SCHEMBL9378264

Cc1ccc(N2N=C(Cn3ccnc3)C(C)C2=O)cc1

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 10/20 0.51
CYP11B1 P15538 7/20 0.51
CYP11B2 P19099 6/20 0.51
LOX P28300 1/20 0.40
LOXL3 P58215 1/20 0.40
LOXL4 Q96JB6 1/20 0.40
LOXL2 Q9Y4K0 1/20 0.40
QPCT Q16769 1/20 0.39
ATM Q13315 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9378886 0.90 CYP19A1 (0.50) CYP19A1CYP11B1CYP11B2QPCT
SCHEMBL9378248 0.90 LOX (0.50) CYP19A1CYP11B1CYP11B2LOXLOXL3
SCHEMBL9383847 0.89 CYP11B1 (0.45) CYP19A1CYP11B1CYP11B2QPCT
SCHEMBL9378661 0.88 CYP19A1 (0.48) CYP19A1CYP11B1CYP11B2ATM
SCHEMBL9378673 0.85 CYP19A1 (0.49) CYP19A1CYP11B1CYP11B2QPCTATM
SCHEMBL9377424 0.85 TBXAS1 (0.42) CYP19A1CYP11B1CYP11B2
SCHEMBL9383432 0.84 CYP19A1 (0.48) CYP19A1CYP11B1CYP11B2QPCTATM
SCHEMBL9382448 0.81 CYP19A1 (0.45) CYP19A1CYP11B1CYP11B2QPCT
SCHEMBL9383526 0.76 CYP19A1 (0.48) CYP19A1CYP11B1CYP11B2
SCHEMBL9378296 0.75 CES2 (0.55) CYP19A1CYP11B1CYP11B2QPCT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0269030-B1 Lipid-peroxide formation inhibiting composition and novel compounds useful therefor MITSUBISHI CHEM IND (JP) 1994-05-04 EP disclosed
US-5089515-A Antiischemic agents; pyrazolone compounds MITSUBISHI KASEI CORPORATION (JP) 1992-02-18 US disclosed
US-4990619-A Cardiovascular disorders, antiischemic agents MITSUBISHI KASEI CORPORATION (JP) 1991-02-05 US disclosed
US-4906644-A Lipid-peroxide formation inhibiting composition and novel compounds useful therefor MITSUBISHI KASEI CORPORATION (JP) 1990-03-06 US disclosed
EP-0269030-A2 Lipid-peroxide formation inhibiting composition and novel compounds useful therefor MITSUBISHI KASEI CORPORATION (JP) 1988-06-01 EP disclosed