SCHEMBL9378296

SCHEMBL9378296

CCC1C(=O)N(c2ccccc2)N=C1Cn1ccnc1

nearest known ligand 0.55

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CES2 O00748 12/20 0.55
CYP19A1 P11511 6/20 0.44
CYP11B1 P15538 4/20 0.44
CYP11B2 P19099 4/20 0.44
CYP1A2 P05177 1/20 0.44
POLB P06746 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
MAPT P10636 1/20 0.44
TBXAS1 P24557 1/20 0.44
QPCT Q16769 1/20 0.44
CYP4Z1 Q86W10 1/20 0.44
QPCTL Q9NXS2 1/20 0.44
CYP17A1 P05093 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9378673 0.90 CYP19A1 (0.49) CES2CYP19A1CYP11B1CYP11B2QPCT
SCHEMBL9380107 0.89 CES2 (0.46) CES2CYP19A1CYP11B1CYP11B2CYP1A2
SCHEMBL9383526 0.88 CYP19A1 (0.48) CES2CYP19A1CYP11B1CYP11B2CYP17A1
SCHEMBL9381460 0.87 CYP19A1 (0.47) CES2CYP19A1CYP11B1CYP11B2
SCHEMBL9379264 0.86 CYP11B1 (0.40) CES2CYP19A1CYP11B1CYP11B2CYP1A2
SCHEMBL9378248 0.85 LOX (0.50) CES2CYP19A1CYP11B1CYP11B2CYP1A2
SCHEMBL9380139 0.84 TBXAS1 (0.41) CES2CYP19A1CYP11B1CYP11B2TBXAS1
SCHEMBL9379529 0.83 SIGMAR1 (0.40) CES2CYP19A1CYP11B1CYP11B2CYP17A1
SCHEMBL9378706 0.82 CYP11B1 (0.43) CES2CYP19A1CYP11B1CYP11B2CYP1A2
SCHEMBL9382448 0.79 CYP19A1 (0.45) CES2CYP19A1CYP11B1CYP11B2QPCT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0269030-B1 Lipid-peroxide formation inhibiting composition and novel compounds useful therefor MITSUBISHI CHEM IND (JP) 1994-05-04 EP disclosed
US-5089515-A Antiischemic agents; pyrazolone compounds MITSUBISHI KASEI CORPORATION (JP) 1992-02-18 US disclosed
US-4906644-A Lipid-peroxide formation inhibiting composition and novel compounds useful therefor MITSUBISHI KASEI CORPORATION (JP) 1990-03-06 US disclosed
EP-0269030-A2 Lipid-peroxide formation inhibiting composition and novel compounds useful therefor MITSUBISHI KASEI CORPORATION (JP) 1988-06-01 EP disclosed