SCHEMBL9384146

SCHEMBL9384146

Cc1ccn2c(=O)c(OC(=O)O)cnc2c1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.64
ALDH1A1 P00352 5/20 0.64
GAA P10253 3/20 0.64
PKM P14618 3/20 0.64
HPGD P15428 3/20 0.57
GLA P06280 1/20 0.57
MAPT P10636 3/20 0.53
NPC1 O15118 4/20 0.46
RAB9A P51151 4/20 0.46
THRB P10828 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.41
HTT P42858 1/20 0.41
HSD17B10 Q99714 1/20 0.39
POLB P06746 2/20 0.39
TP53 P04637 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
GABRG2 P18507 1/20 0.37
GABRB3 P28472 1/20 0.37
GABRA3 P34903 1/20 0.37
CGAS Q8N884 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9387073 0.80 KDM4E (0.55) KDM4EALDH1A1GAAPKMHPGD
SCHEMBL9388014 0.79 KDM4E (0.56) KDM4EALDH1A1GAAPKMHPGD
SCHEMBL9383435 0.79 ALDH1A1 (0.49) KDM4EALDH1A1GAAPKMHPGD
SCHEMBL5717801 0.78 ALDH1A1 (1.00) KDM4EALDH1A1GAAPKMHPGD
SCHEMBL9383229 0.78 ALDH1A1 (0.49) KDM4EALDH1A1GAAPKMHPGD
SCHEMBL22271486 0.76 KDM4E (0.66) KDM4EALDH1A1GAAPKMHPGD
SCHEMBL5912239 0.74 ALDH1A1 (0.76) KDM4EALDH1A1GAAPKMHPGD
SCHEMBL14740159 0.73 KDM4E (0.66) KDM4EALDH1A1GAAPKMHPGD
SCHEMBL9389118 0.72 TP53 (0.50) KDM4EALDH1A1GAAHPGDMAPT
SCHEMBL9382960 0.70 HTT (0.42) KDM4EALDH1A1GAAPKMHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0326981-B1 4-Oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide derivatives, their preparation, medicaments containing them and their preparation CHINOIN GYOGYSZER ES VEGYESZET (HU) 1994-11-09 EP disclosed
EP-0326981-A2 4-Oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide derivatives, their preparation, medicaments containing them and their preparation CHINOIN Gyogyszer és Vegyészeti Termékek Gyára RT. (HU) 1989-08-09 EP disclosed