Sulphamoprine

Sulphamoprine

SCHEMBL93846

COc1cc(OC)nc(NS(=O)(=O)c2ccc(N)cc2)n1

nearest known ligand 0.67

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.67
HTR6 P50406 4/20 0.67
ALDH1A1 P00352 3/20 0.67
CYP3A4 P08684 3/20 0.67
SMN1; SMN2 Q16637 3/20 0.66
TDP1 Q9NUW8 1/20 0.66
TSHR P16473 2/20 0.62
CYP2C19 P33261 3/20 0.61
L3MBTL1 Q9Y468 2/20 0.60
MAPT P10636 4/20 0.56
AURKA O14965 1/20 0.54
DHFR P00374 1/20 0.54
CYP2C9 P11712 2/20 0.54
RAB9A P51151 1/20 0.52
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
KDM4E B2RXH2 1/20 0.51
APEX1 P27695 1/20 0.51
BLM P54132 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Sulphamoprine SCHEMBL2430283 0.98 HTR6 (0.65) LMNAHTR6ALDH1A1CYP3A4SMN1; SMN2
Sulphamoprine SCHEMBL28631928 0.98 HTR6 (0.65) LMNAHTR6ALDH1A1CYP3A4SMN1; SMN2
SCHEMBL17592905 0.92 SMN1; SMN2 (0.76) LMNAHTR6ALDH1A1CYP3A4SMN1; SMN2
SCHEMBL7826186 0.85 HTR6 (0.67) LMNAHTR6ALDH1A1CYP3A4SMN1; SMN2
SCHEMBL2176380 0.84 MAPT (0.68) LMNAHTR6ALDH1A1CYP3A4SMN1; SMN2
SCHEMBL30438514 0.83 LMNA (0.64) LMNAHTR6ALDH1A1CYP3A4SMN1; SMN2
SCHEMBL11882075 0.82 L3MBTL1 (0.77) LMNAHTR6ALDH1A1CYP3A4SMN1; SMN2
SCHEMBL7837632 0.81 HTR6 (0.78) LMNAHTR6ALDH1A1CYP3A4SMN1; SMN2
SCHEMBL31105735 0.81 SMN1; SMN2 (0.54) ALDH1A1SMN1; SMN2TSHRMEN1KMT2A
Sulfametomidine SCHEMBL151238 0.80 HTR6 (0.76) LMNAHTR6ALDH1A1CYP3A4SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 7347 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260091119-A1 ISOLATED TARGETED DELIVERY SYSTEM FOR THE TREATMENT OF GLIOMA CELLIS AG (CH) 2026-04-02 US claimed
US-20260027140-A1 COMPOSITIONS AND METHODS FOR TREATING AND AMELIORATING RESPIRATORY CONDITIONS AND INFLAMMATION OF MUCOSA ATOPIC MEDICAL INC (US) 2026-01-29 US claimed
US-12516365-B2 Biocide compositions compatible with enzyme biosensors and methods of use thereof INSTRUMENTATION LABORATORY COMPANY (US) 2026-01-06 US claimed
US-12465623-B2 Use of parasites and extracellular vesicles obtained from parasites in cancer treatment YEDITEPE UNIVERSITESI (TR) 2025-11-11 US claimed
EP-4637829-A1 ISOLATED TARGETED DELIVERY SYSTEM FOR THE TREATMENT OF OVARIAN CANCER Cellis Sp. z o.o. ([Ltd.] (PL) 2025-10-29 EP claimed
EP-4630043-A1 IMMUNE-ACTIVATING COMPLEXES Dynamic Cell Therapies, Inc. (US) 2025-10-15 EP claimed
EP-4630446-A1 ENGINEERED SWITCHES FOR IMMUNE CELL ACTIVITY AND METHODS OF USE THEREOF Dynamic Cell Therapies, Inc. (US) 2025-10-15 EP claimed
US-20250314664-A1 COMPOSITIONS AND METHODS TO DETECT INFECTIOUS ORGANISMS MARS, INCORPORATED (US) 2025-10-09 US claimed
EP-3965808-B1 USE OF PARASITES AND EXTRACELLULAR VESICLES OBTAINED FROM PARASITES IN CANCER TREATMENT UNIV YEDITEPE (TR) 2025-09-03 EP claimed
EP-4594520-A2 COMPOSITIONS CONTAINING OLIGONUCLEOTIDES WITH THERANOSTIC APPLICATIONS Sixfold Bioscience Ltd. (GB) 2025-08-06 EP claimed
EP-0021847-B1 LONG ACTING SULFONAMIDE INJECTABLE COMPOSITIONS PFIZER INC. (US) 1983-07-20 EP claimed
US-4332796-A MICROCRYSTALS COATED WITH MIXTURES OF PHOSPHOLIPIDS AND NONIONIC SURFACTANTS LABORATORIOS BAGO S.A. (AR) 1982-06-01 US claimed
US-4277248-A FORMATION OF SCHIFF BASE WITH P-DIMETHYLAMINOCINNAMALDEHYDE HOFFMANN-LA ROCHE INC. (US) 1981-07-07 US claimed
EP-0021847-A2 Long acting sulfonamide injectable compositions PFIZER INC. (US) 1981-01-07 EP claimed
US-4169763-A OF A CORYNEBACTERIA RESISTANT TO ASPARTIC ACID ANALOGS AND SULFA DRUGS KYOWA HAKKO KOGYO CO., LTD. (JP) 1979-10-02 US claimed
US-4122158-A FOR TREATMENT OF BURNS; BIODEGRADABLE HYDROPHOBIC POLYMER; SUSTAINED RELEASE ALZA CORPORATION (US) 1978-10-24 US claimed
US-4094976-A ANTICOCCIDIAL CYCLICAMINO ETHANOLS AND ESTERS THEREOF MERCK & CO., INC. (US) 1978-06-13 US claimed
US-4044119-A RUMINANTS, NATIVE MILK SOLIDS, DRUG ENTRAPMENT CUTTER LABORATORIES, INC. (US) 1977-08-23 US claimed
US-4041160-A N-METHYL-2-PYRROLIDONE, ANTICOCCIDIAL AGENTS ABIC LTD. (IL) 1977-08-09 US claimed
US-3983209-A HYDROPHOBIC BIOERODIBLE POLYMER, MICROBIOCIDE OR PROTEOLYTIC ENZYME ALZA CORPORATION (US) 1976-09-28 US claimed