SCHEMBL9387769

SCHEMBL9387769

Sc1c(Cl)cc(Cl)c(Cl)c1S

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.50
HPGD P15428 7/20 0.43
HSD17B10 Q99714 7/20 0.43
TSHR P16473 7/20 0.43
CASP1 P29466 1/20 0.43
ALDH1A1 P00352 2/20 0.40
MAPK1 P28482 3/20 0.39
CRHBP P24387 1/20 0.36
CRHR2 Q13324 1/20 0.36
AHR P35869 9/20 0.36
HSP90AA1 P07900 2/20 0.33
MEN1 O00255 1/20 0.33
NPC1 O15118 1/20 0.33
USP2 O75604 1/20 0.33
EGFR P00533 1/20 0.33
LMNA P02545 1/20 0.33
ESR1 P03372 1/20 0.33
ERBB2 P04626 1/20 0.33
CYP1A2 P05177 1/20 0.33
LCK P06239 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9357749 1.00 CYP3A4 (0.50) CYP3A4HPGDHSD17B10TSHRCASP1
SCHEMBL48326 0.87 CYP3A4 (0.56) CYP3A4HPGDHSD17B10TSHRCASP1
SCHEMBL6520758 0.81 CYP3A4 (0.59) CYP3A4HPGDHSD17B10TSHRCASP1
SCHEMBL6512985 0.79 CYP3A4 (0.56) CYP3A4HPGDHSD17B10TSHRCASP1
SCHEMBL6512992 0.79 CYP3A4 (0.56) CYP3A4HPGDHSD17B10TSHRCASP1
SCHEMBL6511604 0.79 CYP3A4 (0.56) CYP3A4HPGDHSD17B10TSHRCASP1
SCHEMBL9480774 0.73 CYP3A4 (0.40) CYP3A4HPGDHSD17B10TSHRCASP1
SCHEMBL16312908 0.69 CYP3A4 (0.38) CYP3A4HPGDHSD17B10TSHRCASP1
Pentachlorobenzene SCHEMBL11455164 0.68 CYP3A4 (1.00) CYP3A4HPGDHSD17B10TSHRCASP1
Pentachlorobenzene SCHEMBL183144 0.68 CYP3A4 (1.00) CYP3A4HPGDHSD17B10TSHRCASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-58105960-A None JP disclosed
JP-6025151-A None JP disclosed
JP-H0625151-A PRODUCTION OF O-BENZENEDITHIOL COMPOUND MITSUI TOATSU CHEM INC 1994-02-01 JP disclosed
US-4508655-A NEAR INFRARED ABSORBERS MITSUI TOATSU CHEMICALS, INC. (JP) 1985-04-02 US disclosed
JP-S58105960-A NOVEL HALOGEN-SUBSTITUTED O-BENZENEDITHIOL AND ITS PREPARATION MITSUI TOATSU CHEM INC 1983-06-24 JP disclosed