SCHEMBL9389330

SCHEMBL9389330

N#Cc1cccc2c(=O)cc(O)c(=O)[nH]c12

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
DAO P14920 8/20 0.42
DDO Q99489 5/20 0.42
PLA2G7 Q13093 3/20 0.41
MCL1 Q07820 2/20 0.41
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
AR P10275 1/20 0.38
FASN P49327 2/20 0.38
UPP1 Q16831 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9387820 0.81 UPP1 (0.39) KDM4ETDP1DAODDOMCL1
SCHEMBL9389836 0.78 UPP1 (0.42) KDM4EDAODDOMCL1FASN
SCHEMBL9389395 0.76 KDM4E (0.46) KDM4ETDP1DAODDOPLA2G7
SCHEMBL9389416 0.76 DAO (0.66) KDM4ETDP1DAODDOPLA2G7
SCHEMBL8583717 0.76 DAO (0.66) KDM4ETDP1DAODDOPLA2G7
SCHEMBL9388997 0.76 DAO (0.66) KDM4ETDP1DAODDOPLA2G7
SCHEMBL9393346 0.76 DAO (0.49) KDM4ETDP1DAODDOPLA2G7
SCHEMBL3358803 0.76 FASN (0.40) KDM4EDAODDOMCL1CA1
SCHEMBL9389922 0.76 DAO (0.46) DAODDOMCL1FASNUPP1
SCHEMBL9389937 0.76 FASN (0.35) DAODDOMCL1FASNUPP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1994007500-A1 2,5-DIHYDRO-2,5-DIOXO-1H-AZEPINES AND 2,5-DIHYDRO-2-OXO-1H-AZEPINES AND THE USE THEREOF AS EXCITATORY AMINO ACID AND GLYCINE RECEPTOR ANTAGONISTS WEBER ECKARD (US) 1994-04-14 WO disclosed