SCHEMBL9392647

SCHEMBL9392647

N#Cc1ccc2c(=O)cc(O)c(=O)[nH]c2c1

nearest known ligand 0.56

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
FASN P49327 1/20 0.47
NOS3 P29474 1/20 0.43
NOS1 P29475 1/20 0.43
NOS2 P35228 1/20 0.43
AR P10275 1/20 0.42
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
DAO P14920 4/20 0.41
DDO Q99489 3/20 0.41
SERPINE1 P05121 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9393317 0.88 FASN (0.57) FASNARCA1CA2DAO
SCHEMBL3396789 0.81 DAO (0.63) FASNNOS3NOS1NOS2DAO
SCHEMBL9387738 0.79 DAO (0.65) DAODDO
SCHEMBL9007832 0.76 DAO (0.65) DAODDO
SCHEMBL9007836 0.76 METAP2 (0.49) DAODDO
SCHEMBL7350621 0.76 DAO (0.65) DAO
SCHEMBL3363129 0.75 DAO (0.54) FASNDAODDO
SCHEMBL3422876 0.75 DAO (0.54) FASNDAODDO
SCHEMBL25246466 0.74 PARP1 (0.56) FASNNOS3NOS1NOS2CA1
SCHEMBL9393132 0.74 GRIN2D (0.38) FASNDAODDO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1994007500-A1 2,5-DIHYDRO-2,5-DIOXO-1H-AZEPINES AND 2,5-DIHYDRO-2-OXO-1H-AZEPINES AND THE USE THEREOF AS EXCITATORY AMINO ACID AND GLYCINE RECEPTOR ANTAGONISTS WEBER ECKARD (US) 1994-04-14 WO disclosed