SCHEMBL9393145

SCHEMBL9393145

Cc1ccc2c(=O)c(O)cc(=O)[nH]c2c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.53
ALDH1A1 P00352 2/20 0.53
GLA P06280 2/20 0.53
GAA P10253 2/20 0.53
HPGD P15428 1/20 0.53
DAO P14920 2/20 0.47
DDO Q99489 1/20 0.47
LMNA P02545 1/20 0.46
TP53 P04637 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
KIF11 P52732 2/20 0.44
EGFR P00533 1/20 0.44
MEN1 O00255 1/20 0.44
NPC1 O15118 1/20 0.44
POLB P06746 1/20 0.44
KMT2A Q03164 1/20 0.44
CA12 O43570 1/20 0.43
CA9 Q16790 1/20 0.43
MPL P40238 1/20 0.43
KDM5A P29375 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8109985 0.89 KDM4E (0.59) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL8581212 0.82 KDM4E (0.66) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL2795205 0.80 KDM4E (0.67) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL9393238 0.79 KDM4E (0.47) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL2272868 0.79 ALDH1A1 (0.59) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL31081977 0.79 ALDH1A1 (0.59) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL9388988 0.77 KDM4E (0.79) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL9392742 0.76 DAO (0.52) KDM4EALDH1A1HPGDDAODDO
SCHEMBL9571854 0.76 MEN1 (0.65) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL9155186 0.76 ALDH1A1 (0.45) KDM4EALDH1A1GLAGAAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1994007500-A1 2,5-DIHYDRO-2,5-DIOXO-1H-AZEPINES AND 2,5-DIHYDRO-2-OXO-1H-AZEPINES AND THE USE THEREOF AS EXCITATORY AMINO ACID AND GLYCINE RECEPTOR ANTAGONISTS WEBER ECKARD (US) 1994-04-14 WO disclosed