SCHEMBL939617

SCHEMBL939617

O=C(/C=C\C(=O)OC(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)F)OC(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)F

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.39
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30
MMP1 P03956 1/20 0.30
MMP2 P08253 1/20 0.30
MMP9 P14780 1/20 0.30
MMP8 P22894 1/20 0.30
MMP13 P45452 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1426649 1.00 THRB (0.39) THRBCA1CA2MMP1MMP2
SCHEMBL1902943 1.00 THRB (0.39) THRBCA1CA2MMP1MMP2
SCHEMBL11862837 1.00 THRB (0.39) THRBCA1CA2MMP1MMP2
SCHEMBL1426813 1.00 THRB (0.39) THRBCA1CA2MMP1MMP2
SCHEMBL28705529 0.98 THRB (0.36) THRB
SCHEMBL5704591 0.92 HCAR2 (0.39) THRB
SCHEMBL1536821 0.83 THRB (0.37) THRB
SCHEMBL1537075 0.83 THRB (0.37) THRB
SCHEMBL534358 0.83 THRB (0.37) THRB
SCHEMBL528801 0.83 THRB (0.37) THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 44 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1455663-A Novel aerosol formulation containing polar fluorinated molecule ASTRAZENECA AB (SE) 2003-11-12 CN claimed
US-9720339-B2 Toner, developer using the toner, image forming apparatus RICOH COMPANY, LTD. (JP) 2017-08-01 US disclosed
EP-2813895-B1 Toner, Developer, and Image Forming Apparatus RICOH CO LTD (JP) 2017-07-05 EP disclosed
EP-2769266-B1 TONER, DEVELOPER USING THE TONER, IMAGE FORMING APPARATUS RICOH CO LTD (JP) 2017-01-11 EP disclosed
US-9519235-B2 Toner, developer using the toner, image forming apparatus RICOH COMPANY, LTD. (JP) 2016-12-13 US disclosed
US-20160334726-A1 TONER, DEVELOPER USING THE TONER, IMAGE FORMING APPARATUS SAKASHITA SHINGO (JP) 2016-11-17 US disclosed
US-9366982-B2 Toner, developer, and image forming apparatus RICOH COMPANY, LTD. (JP) 2016-06-14 US disclosed
US-9134638-B2 Toner, developer using the toner, image forming apparatus RICOH COMPANY, LTD. (JP) 2015-09-15 US disclosed
US-20150227071-A1 TONER, DEVELOPER USING THE TONER, IMAGE FORMING APPARATUS SAKASHITA SHINGO (JP) 2015-08-13 US disclosed
EP-2813895-A1 Toner, Developer, and Image Forming Apparatus Ricoh Company, Ltd. (JP) 2014-12-17 EP disclosed
US-20070218390-A1 TONER FOR DEVELOPING ELECTROSTATIC IMAGES, PRODUCTION METHOD THEREOF; DEVELOPER, IMAGE FORMING METHOD, IMAGE FORMING APPARATUS, AND PROCESS CARTRIDGE RICOH COMPANY LTD. (JP) 2007-09-20 US disclosed
US-20070218393-A1 TONER FOR DEVELOPING ELECTROSTATIC IMAGE, AND DEVELOPER, TONER CONTAINER, IMAGE FORMING APPARATUS AND PROCESS CARTRIDGE USING THE TONER RICOH COMPANY, LIMITED (JP) 2007-09-20 US disclosed
US-20070190442-A1 TONER, AND DEVELOPER, IMAGE FORMING METHOD, IMAGE FORMING APPARATUS, AND PROCESS CARTRIDGE USING THE TONER RICOH COMPANY, LTD. (JP) 2007-08-16 US disclosed
US-20070166635-A1 TONER AND METHOD OF PREPARING THE TONER RICOH COMPANY LIMITED (JP) 2007-07-19 US disclosed
US-20060204882-A1 Toner, toner manufacturing method, developer, image forming apparatus, and process cartridge for the image forming apparatus RICOH COMPANY LIMITED (JP) 2006-09-14 US disclosed
WO-2003102685-A9 METHODS OF SURFACE MODIFICATION FOR IMPROVING ELECTROPHORETIC DISLAY PERFORMANCE SIPIX IMAGING INC (US) 2004-02-19 WO disclosed
WO-2003102685-A2 METHODS OF SURFACE MODIFICATION FOR IMPROVING ELECTROPHORETIC DISLAY PERFORMANCE SIPIX IMAGING, INC. (US) 2003-12-11 WO disclosed
US-20030210455-A1 Methods of surface modification for improving electrophoretic display performance E INK CALIFORNIA, LLC 2003-11-13 US disclosed
CN-1455663-A Novel aerosol formulation containing polar fluorinated molecule ASTRAZENECA AB (SE) 2003-11-12 CN disclosed
US-6303730-B1 NONHYDROLYTIC CONDENSATION OF CHLOROSILANES WITH POLYMERIZABLE GROUPS AND OPTIONALLY FLUORINATED GROUPS, WITH THE HELP OF A CONDENSATION AGENT AND THERMAL AND/OR PHOTOCHEMICAL POLYMERIZATION OF THE OBTAINED CONDENSATION PRODUCT INSTITUT FUR NEUE MATERIALIEN GEMEINNUTZIGE GMBH (DE) 2001-10-16 US disclosed