SCHEMBL9396641

SCHEMBL9396641

O=S(=O)(NCBr)c1ccccc1-c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 2/20 0.48
EDNRA P25101 5/20 0.46
EDNRB P24530 4/20 0.46
CCR1 P32246 1/20 0.41
FEN1 P39748 4/20 0.41
ALOX5AP P20292 2/20 0.41
UCHL1 P09936 1/20 0.41
USP30 Q70CQ3 1/20 0.41
BCL2 P10415 1/20 0.40
BCL2L1 Q07817 1/20 0.40
MCL1 Q07820 1/20 0.40
BCL2A1 Q16548 1/20 0.40
BCL2L2 Q92843 1/20 0.40
OPRM1 P35372 1/20 0.40
OPRK1 P41145 1/20 0.40
FBP1 P09467 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30517195 0.78 EDNRA (0.45) CASP1EDNRAEDNRBCCR1FEN1
SCHEMBL29537027 0.77 CA2 (0.58) CASP1EDNRAEDNRBUCHL1USP30
SCHEMBL1767981 0.77 CA2 (0.58) CASP1EDNRAEDNRBUCHL1USP30
SCHEMBL3632239 0.77 CA12 (0.62) EDNRAEDNRBCCR1
SCHEMBL2006242 0.77 PKLR (0.56) CASP1CCR1
SCHEMBL15924985 0.76 FEN1 (0.55) CASP1CCR1FEN1ALOX5AP
SCHEMBL1846856 0.76 CASP1 (0.51) CASP1EDNRAEDNRBFEN1ALOX5AP
SCHEMBL10780146 0.76 CASP1 (0.51) CASP1EDNRAEDNRBFEN1ALOX5AP
SCHEMBL15668311 0.76 CASP1 (0.51) CASP1EDNRAEDNRBFEN1ALOX5AP
SCHEMBL418847 0.76 CASP1 (0.51) CASP1EDNRAEDNRBFEN1ALOX5AP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5292741-A Macrocycles incorporating quinazolinones MERCK & CO., INC. (US) 1994-03-08 US disclosed
US-5262412-A Angiotensin II antagonists, hypotensive agents, treatment of congestive heart failure and glaucoma MERCK & CO., INC. (US) 1993-11-16 US disclosed