SCHEMBL9397258

SCHEMBL9397258

Clc1cccc(CCN2CCNCC2)c1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 8/20 0.65
SLC6A4 P31645 4/20 0.59
SLC6A2 P23975 2/20 0.52
SLC6A3 Q01959 2/20 0.52
KCNH2 Q12809 1/20 0.52
HTR6 P50406 3/20 0.52
KDM4E B2RXH2 1/20 0.51
ALDH1A1 P00352 1/20 0.51
HTR2C P28335 2/20 0.51
CYP2C9 P11712 2/20 0.50
CYP2C19 P33261 2/20 0.50
HTR3E A5X5Y0 1/20 0.50
HTR3B O95264 1/20 0.50
TP53 P04637 1/20 0.50
CYP1A2 P05177 1/20 0.50
ADRB1 P08588 1/20 0.50
CYP3A4 P08684 1/20 0.50
HTR1A P08908 1/20 0.50
CYP2D6 P10635 1/20 0.50
THRB P10828 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9398424 0.94 SIGMAR1 (0.68) SIGMAR1SLC6A4SLC6A2SLC6A3KCNH2
SCHEMBL10643080 0.91 SIGMAR1 (0.67) SIGMAR1SLC6A4SLC6A2SLC6A3HTR6
SCHEMBL2256688 0.88 SIGMAR1 (0.59) SIGMAR1SLC6A4SLC6A2KCNH2KDM4E
SCHEMBL1888148 0.83 SIGMAR1 (0.72) SIGMAR1SLC6A4SLC6A2HTR6KDM4E
SCHEMBL29478520 0.83 SIGMAR1 (0.72) SIGMAR1SLC6A4SLC6A2HTR6KDM4E
Hydrochloric Acid SCHEMBL4819656 0.82 SIGMAR1 (0.70) SIGMAR1HTR6KDM4EALDH1A1CYP2C9
SCHEMBL28742033 0.82 SIGMAR1 (0.56) SIGMAR1SLC6A4SLC6A3HTR1AHRH3
SCHEMBL8411258 0.81 SLC6A3 (0.73) SIGMAR1SLC6A4SLC6A2SLC6A3KCNH2
SCHEMBL12879708 0.81 HRH3 (0.73) SIGMAR1SLC6A4SLC6A2SLC6A3KCNH2
SCHEMBL9397221 0.81 SIGMAR1 (0.56) SIGMAR1SLC6A4SLC6A3HTR1AHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5340811-A Bronchodilator agent ASAHI KASEI KOGYO KABUSHIKI KAISHA (JP) 1994-08-23 US disclosed
EP-0250361-B1 Disubstituted piperazines CIBA GEIGY AG (CH) 1993-12-08 EP disclosed
EP-0471841-A1 SULFONAMIDE DERIVATIVE AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME Asahi Kasei Kogyo Kabushiki Kaisha (JP) 1992-02-26 EP disclosed
US-4804661-A ANALGESICS CIBA-GEIGY CORPORATION (US) 1989-02-14 US disclosed
EP-0250361-A2 Disubstituted piperazines CIBA-GEIGY AG (CH) 1987-12-23 EP disclosed