Dropropizine

Dropropizine

SCHEMBL93975

OCC(O)CN1CCN(c2ccccc2)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 1/20 1.00
ADRA2B P18089 1/20 1.00
ADRA2C P18825 1/20 1.00
KMT2A Q03164 3/20 0.66
MEN1 O00255 2/20 0.66
MAPT P10636 5/20 0.64
TSHR P16473 1/20 0.62
IGF1R P08069 1/20 0.57
MAPK1 P28482 2/20 0.57
L3MBTL1 Q9Y468 2/20 0.57
KDM4E B2RXH2 2/20 0.57
ALDH1A1 P00352 2/20 0.57
GAA P10253 1/20 0.57
GFER P55789 1/20 0.57
TDP1 Q9NUW8 1/20 0.56
ADRA1B P35368 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Dropropizine SCHEMBL8379428 1.00 ADRA2A (1.00) ADRA2AADRA2BADRA2CKMT2AMEN1
Levodropropizine SCHEMBL29043 1.00 ADRA2A (1.00) ADRA2AADRA2BADRA2CKMT2AMEN1
Dropropizine SCHEMBL27495915 0.98 ADRA2A (0.97) ADRA2AADRA2BADRA2CKMT2AMEN1
Dropropizine SCHEMBL10445730 0.91 ADRA2A (0.83) ADRA2AADRA2BADRA2CKMT2AMEN1
Dropropizine SCHEMBL10445733 0.90 ADRA2A (0.81) ADRA2AADRA2BADRA2CKMT2AMEN1
Dropropizine SCHEMBL10445975 0.90 ADRA2A (0.81) ADRA2AADRA2BADRA2CKMT2AMEN1
Dropropizine SCHEMBL10446140 0.90 ADRA2A (0.81) ADRA2AADRA2BADRA2CKMT2AMEN1
Dropropizine SCHEMBL10446134 0.90 ADRA2A (0.81) ADRA2AADRA2BADRA2CKMT2AMEN1
Dropropizine SCHEMBL10445732 0.90 ADRA2A (0.81) ADRA2AADRA2BADRA2CKMT2AMEN1
Dropropizine SCHEMBL10445734 0.85 ADRA2A (0.72) ADRA2AADRA2BADRA2CKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 802 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250255781-A1 PROCESSES FOR PREPARATION OF 3-D PRINTED PHARMACEUTICAL PRODUCTS BRISTOL-MYERS SQUIBB COMPANY (US) 2025-08-14 US claimed
US-12296043-B2 Liquisoft capsules PATHEON SOFTGELS INC. (US) 2025-05-13 US claimed
EP-4510999-A1 PROCESSES FOR PREPARATION OF 3-D PRINTED PHARMACEUTICAL PRODUCTS Bristol-Myers Squibb Company (US) 2025-02-26 EP claimed
US-20240165020-A1 LIQUISOFT CAPSULES PATHEON SOFTGELS INC (US) 2024-05-23 US claimed
EP-4360653-A2 LIQUISOFT CAPSULES Patheon Softgels Inc. (US) 2024-05-01 EP claimed
US-20240082176-A1 DROPROPIZINE IN COMBINATION WITH AMBROXOL IN THE DOSAGE FORM OF SYRUP AND TABLETS PRODUCTOS FARMACEUTICOS, S.A. DE C.V. (MX) 2024-03-14 US claimed
US-11872307-B2 Liquisoft capsules PATHEON SOFTGELS INC. (US) 2024-01-16 US claimed
EP-3682872-B1 LIQUISOFT CAPSULES PATHEON SOFTGELS INC (US) 2024-01-03 EP claimed
US-20230414575-A1 MK2 ACTIVATING COMPOUNDS FOR USE IN TREATING VASCULAR LEAK AND ENDOTHELIAL BARRIER DISORDERS AKTTYVA THERAPEUTICS INC (US) 2023-12-28 US claimed
WO-2023205619-A1 PROCESSES FOR PREPARATION OF 3-D PRINTED PHARMACEUTICAL PRODUCTS BRISTOL-MYERS SQUIBB COMPANY (US) 2023-10-26 WO claimed
WO-1994020449-A1 SALTS OF 2-(3-BENZOYLPHENYL)PROPIONIC ACID WITH ACHIRAL AND CHIRAL ORGANIC BASES AND PHARMACEUTICAL COMPOSITIONS THEREOF DOMPE'FARMACEUTICI SPA (IT) 1994-09-15 WO claimed
US-5087698-A Using L(+)tartaric acid DOMPE' FARMACEUTICI S.P.A. (IT) 1992-02-11 US claimed
EP-0409044-A2 A process for the optical resolution of dropropizine DOMPE' FARMACEUTICI S.p.A. (IT) 1991-01-23 EP claimed
EP-0147847-B1 OPTICALLY ACTIVE COMPOUNDS WITH ANTITUSSIVE AND CENTRAL SEDATIVE ACTIVITY, A PROCESS FOR THE PREPARATION THEREOF AND COMPOSITIONS CONTAINING THE SAME DOMPE' FARMACEUTICI S.p.A. (IT) 1990-03-07 EP claimed
EP-0349066-A1 Preparation of enantiomers of dropropizine DSM N.V. (NL) 1990-01-03 EP claimed
EP-0348713-A1 (R,S)-3-(4-phenyl-1-piperazinyl)-1,2-propanediol salts DOTT. FORMENTI S.P.A. INDUSTRIA CHIMICA E FARMACEUTICA (IT) 1990-01-03 EP claimed
US-4764515-A REDUCED SIDE EFFECTS DOMPE' FARMACEUTICI S.P.A. (IT) 1988-08-16 US claimed
US-4699911-A Levo and dextro dropropizine having antitussive activity DOMPE' FARMACEUTICI S.P.A. (IT) 1987-10-13 US claimed
EP-0156331-A2 Benzofuran derivatives, processes for preparing the same and antihypertensive agents containing the same KAKEN PHARMACEUTICAL CO., LTD. (JP) 1985-10-02 EP claimed
EP-0147847-A2 Optically active compounds with antitussive and central sedative activity, a process for the preparation thereof and compositions containing the same DOMPE' FARMACEUTICI S.p.A. (IT) 1985-07-10 EP claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240082176-A1 DROPROPIZINE IN COMBINATION WITH AMBROXOL IN THE DOSAGE FORM OF SYRUP AND TABLETS QDPR, IL5, CYP3A5 ADRA2A 186/4885ADRA2B 271/4885ADRA2C 51/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.