SCHEMBL9401009

SCHEMBL9401009

CCOC(=O)N1CCN(c2ncc(-c3cccc(C(F)(F)F)c3)cn2)CC1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.59
HPGD P15428 4/20 0.58
SMN1; SMN2 Q16637 3/20 0.58
MEN1 O00255 7/20 0.58
KMT2A Q03164 7/20 0.58
SLC6A7 Q99884 1/20 0.57
MAPT P10636 3/20 0.54
NPSR1 Q6W5P4 2/20 0.54
KDM4E B2RXH2 1/20 0.54
RAB9A P51151 2/20 0.52
NPC1 O15118 1/20 0.52
GRIN2B Q13224 4/20 0.50
LMNA P02545 2/20 0.50
MAPK1 P28482 2/20 0.50
GRIN1 Q05586 2/20 0.50
ALOX15 P16050 2/20 0.50
HTT P42858 2/20 0.49
USP2 O75604 1/20 0.49
CYP1A2 P05177 2/20 0.49
CYP2C9 P11712 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9400930 0.84 SMN1; SMN2 (0.71) ALDH1A1HPGDSMN1; SMN2MEN1KMT2A
SCHEMBL9400885 0.83 KMT2A (0.62) ALDH1A1SMN1; SMN2MEN1KMT2AMAPT
SCHEMBL593921 0.83 SMN1; SMN2 (0.64) ALDH1A1HPGDSMN1; SMN2MEN1KMT2A
SCHEMBL595155 0.78 ALDH1A1 (0.55) ALDH1A1HPGDSMN1; SMN2MEN1KMT2A
SCHEMBL9401018 0.77 GAK (0.66) ALDH1A1SMN1; SMN2MEN1KMT2AMAPT
SCHEMBL5238917 0.77 SMN1; SMN2 (0.56) ALDH1A1HPGDSMN1; SMN2MEN1KMT2A
SCHEMBL593375 0.77 SMN1; SMN2 (0.56) ALDH1A1HPGDSMN1; SMN2MEN1KMT2A
SCHEMBL11362502 0.76 AOC3 (0.77)
SCHEMBL9400866 0.76 MAPT (0.58) ALDH1A1HPGDSMN1; SMN2MEN1KMT2A
SCHEMBL10373050 0.76 SLC6A7 (0.46) ALDH1A1SLC6A7KDM4EGRIN2BLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5314884-A Antidepressants, anxiolytic agents TROPONWERKE GMBH & CO. (DE) 1994-05-24 US disclosed
US-5187276-A Anxiolytics, neuroleptics, antidepressants, and nootropic agents TROPONWERKE GMBH & CO. KG. (DE) 1993-02-16 US disclosed
US-4988809-A CENTRAL NERVOUS SYSTEM TROPONWERKE GMBH & CO., KG (DE) 1991-01-29 US disclosed
EP-0129128-B1 2-PYRIMIDINYL-1-PIPERAZINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND MEDICINES CONTAINING THEM Troponwerke GmbH & Co. KG (DE) 1990-11-22 EP disclosed
US-4937343-A NEUROLEPTICS OR ANTIDEPRESSANTS TROPONWERKE GMBH & CO. KG (DE) 1990-06-26 US disclosed
US-4818756-A CENTRAL NERVOUS SYSTEM DISORDERS TROPONWERKE GMBH & CO., KG (DE) 1989-04-04 US disclosed