SCHEMBL9401663

SCHEMBL9401663

COC(=O)C1=C(C)NC(C)=C(C(=O)O)C1c1cccc2ccccc12

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.58
HSD17B10 Q99714 6/20 0.58
KMT2A Q03164 5/20 0.58
CYP2C9 P11712 4/20 0.58
ADORA3 P0DMS8 4/20 0.58
CYP1A2 P05177 4/20 0.58
ALDH1A1 P00352 4/20 0.58
MAPT P10636 4/20 0.58
ABCB11 O95342 4/20 0.58
LMNA P02545 4/20 0.58
CACNA1F O60840 4/20 0.58
CACNA1D Q01668 4/20 0.58
CACNA1S Q13698 4/20 0.58
CACNA1C Q13936 4/20 0.58
CYP3A4 P08684 3/20 0.58
CYP2C19 P33261 3/20 0.58
HIF1A Q16665 3/20 0.58
SCN1A P35498 3/20 0.58
SCN5A Q14524 3/20 0.58
SCN2A Q99250 3/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3059360 0.95 KDM4E (0.64) KDM4EHSD17B10KMT2ACYP2C9ADORA3
SCHEMBL3049870 0.91 KMT2A (0.49) KDM4EHSD17B10KMT2ACYP2C9ADORA3
SCHEMBL11829270 0.88 CYP2C9 (0.67) KDM4EHSD17B10KMT2ACYP2C9ADORA3
SCHEMBL11004464 0.82 CYP1A2 (0.68) KDM4EHSD17B10KMT2ACYP2C9ADORA3
SCHEMBL11004457 0.82 CYP1A2 (0.68) KDM4EHSD17B10KMT2ACYP2C9ADORA3
SCHEMBL3034993 0.82 ADORA3 (0.57) KDM4EHSD17B10KMT2ACYP2C9ADORA3
SCHEMBL3026759 0.82 KDM4E (0.62) KDM4EHSD17B10KMT2ACYP2C9ADORA3
SCHEMBL2996737 0.82 MAPT (0.70) KDM4EHSD17B10KMT2ACYP2C9ADORA3
SCHEMBL7414856 0.82 NR1I2 (0.67) KDM4EHSD17B10KMT2ACYP2C9ADORA3
SCHEMBL9830577 0.81 CACNA1B (0.63) KMT2AADORA3CACNA1CCACNA1BMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5286869-A Vasodilators and anticoagulants FUJIREBIO KABUSHIKI KAISHA (JP) 1994-02-15 US disclosed
EP-0403957-A2 Optical active 1,4-dihydropyridine derivates FUJIREBIO INC. (JP) 1990-12-27 EP disclosed
US-4532248-A Administering 1,4-dihydropyridine derivative exhibiting positive inotropic activity BAYER AKTIENGESELLSCHAFT (DE) 1985-07-30 US disclosed