SCHEMBL9401720

SCHEMBL9401720

COC(=O)C1=C(C)NC(C)=C(C(=O)O)C1c1ccoc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 1/20 0.64
ADORA3 P0DMS8 1/20 0.53
TSHR P16473 4/20 0.52
KDM4E B2RXH2 6/20 0.51
HSD17B10 Q99714 4/20 0.51
ALDH1A1 P00352 4/20 0.51
HTT P42858 3/20 0.51
RAB9A P51151 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
MAPT P10636 3/20 0.50
HPGD P15428 2/20 0.50
KMT2A Q03164 2/20 0.50
GAA P10253 1/20 0.50
POLB P06746 2/20 0.49
CACNA1F O60840 1/20 0.49
CACNA1D Q01668 1/20 0.49
CACNA1S Q13698 1/20 0.49
CACNA1C Q13936 1/20 0.49
MEN1 O00255 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27566517 0.90 CACNA1B (0.62) CACNA1BADORA2BCYP1A2CYP2C9MAPK1
SCHEMBL6951320 0.81 ADORA3 (0.76) CACNA1BADORA3TSHRKDM4EHSD17B10
SCHEMBL3010290 0.81 ADORA2B (0.67) CACNA1BADORA3TSHRKDM4EHSD17B10
SCHEMBL7265410 0.80 TSHR (0.65) CACNA1BADORA3TSHRKDM4EHSD17B10
SCHEMBL27520045 0.80 CACNA1B (0.65) CACNA1BTSHRKDM4EHSD17B10ALDH1A1
SCHEMBL7158395 0.79 ADORA3 (0.60) CACNA1BADORA3TSHRKDM4EHSD17B10
SCHEMBL5857481 0.78 CACNA1B (1.00) CACNA1B
SCHEMBL5857475 0.78 CACNA1B (1.00) CACNA1B
SCHEMBL9401767 0.78 KDM4E (0.68) ADORA3TSHRKDM4EHSD17B10ALDH1A1
SCHEMBL9272854 0.78 CACNA1F (0.69) CACNA1BADORA3TSHRKDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5286869-A Vasodilators and anticoagulants FUJIREBIO KABUSHIKI KAISHA (JP) 1994-02-15 US disclosed
EP-0403957-A2 Optical active 1,4-dihydropyridine derivates FUJIREBIO INC. (JP) 1990-12-27 EP disclosed