SCHEMBL9402014

SCHEMBL9402014

Cc1nc2ccccc2c(=O)n1Cc1ccc(-c2ccccc2-c2nnnn2C(c2ccccc2)(c2ccccc2)c2ccccc2)cc1

nearest known ligand 0.57

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 1/20 0.57
AGTR2 P50052 1/20 0.57
AGT P01019 2/20 0.52
ALDH1A1 P00352 4/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
HDAC1 Q13547 1/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
RAB9A P51151 2/20 0.45
LMNA P02545 1/20 0.45
RECQL P46063 1/20 0.45
CYP1A2 P05177 1/20 0.43
GAA P10253 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
TSHR P16473 1/20 0.43
GFER P55789 1/20 0.43
POLB P06746 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9402029 0.90 AGTR1 (0.59) AGTR1AGTR2AGTALDH1A1MEN1
SCHEMBL9402070 0.89 AGTR1 (0.54) AGTR1AGTR2AGTALDH1A1MEN1
SCHEMBL9402017 0.88 AGTR1 (0.69) AGTR1AGTR2AGT
SCHEMBL9402064 0.88 AGTR1 (0.55) AGTR1AGTR2AGTALDH1A1MEN1
SCHEMBL9402043 0.87 AGTR1 (0.55) AGTR1AGTR2AGTALDH1A1MEN1
SCHEMBL9851456 0.86 AGTR1 (0.52) AGTR1AGTR2AGTLMNAPOLB
SCHEMBL9265478 0.83 AGTR1 (0.56) AGTR1AGTR2AGTALDH1A1MEN1
SCHEMBL9263837 0.81 AGT (0.57) AGTR1AGTR2AGT
SCHEMBL9851445 0.79 AGTR1 (0.53) AGTR1AGTR2AGTSMN1; SMN2RAB9A
SCHEMBL13679193 0.78 AGTR1 (0.55) AGTR1AGTR2AGTALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5304565-A Angiotensin II antagonists TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-04-19 US disclosed
EP-0445811-A2 Nitrogen-containing heterocyclic compounds, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-09-11 EP disclosed