SCHEMBL9403359

SCHEMBL9403359

C=C(CC(=O)NCc1ccccc1)C(=O)OC(N)c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.47
MAPT P10636 1/20 0.47
GAA P10253 1/20 0.44
KMT2A Q03164 4/20 0.43
HPGD P15428 2/20 0.43
MEN1 O00255 3/20 0.43
SLC1A1 P43005 1/20 0.42
CRHBP P24387 1/20 0.42
CRHR2 Q13324 1/20 0.42
TSHR P16473 1/20 0.42
RECQL P46063 1/20 0.42
NPSR1 Q6W5P4 1/20 0.41
MCL1 Q07820 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
HTT P42858 1/20 0.40
LMNA P02545 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10690766 0.83 ALDH1A1 (0.55) ALDH1A1MAPTGAAKMT2AHPGD
SCHEMBL7500457 0.82 ALDH1A1 (0.49) ALDH1A1MAPTGAAKMT2AHPGD
SCHEMBL12479803 0.82 CYP19A1 (0.51) ALDH1A1MAPTTSHR
SCHEMBL5176551 0.75 GAA (0.56) ALDH1A1MAPTGAAKMT2AHPGD
SCHEMBL5176559 0.75 GAA (0.59) ALDH1A1MAPTGAAKMT2AHPGD
SCHEMBL9403358 0.74 GAA (0.58) ALDH1A1MAPTGAAKMT2AHPGD
SCHEMBL7802681 0.72 ALDH1A1 (0.57) ALDH1A1MAPTKMT2AMEN1LMNA
SCHEMBL3087061 0.71 GAA (0.73) ALDH1A1MAPTGAAKMT2AHPGD
SCHEMBL8013057 0.70 HPGD (0.44) ALDH1A1KMT2AHPGDTSHRLMNA
SCHEMBL4220537 0.70 KMT2A (0.55) GAAKMT2AMEN1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5321139-A Amination of phenylitaconic anhydride, catalytic reduction of formed amide; renin inhibitor HOECHST AKTIENGESELLSCHAFT (DE) 1994-06-14 US disclosed