SCHEMBL9404233

SCHEMBL9404233

CN1CCN(c2nc(Cl)nc3cccc(C(F)(F)F)c23)CC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 8/20 0.51
CYP1A2 P05177 5/20 0.51
CYP3A4 P08684 5/20 0.51
CYP2D6 P10635 5/20 0.51
MAPK1 P28482 2/20 0.51
HTR3B O95264 4/20 0.48
HTR3A P46098 4/20 0.48
CYP2C19 P33261 4/20 0.47
SMN1; SMN2 Q16637 2/20 0.44
TSHR P16473 3/20 0.42
ALDH1A1 P00352 2/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
CNR2 P34972 1/20 0.42
USP2 O75604 1/20 0.42
HIF1A Q16665 1/20 0.42
KDM4E B2RXH2 2/20 0.42
HSD17B10 Q99714 2/20 0.42
TDP1 Q9NUW8 1/20 0.42
HTR3E A5X5Y0 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9404529 0.85 CYP1A2 (0.51) CYP1A2CYP3A4CYP2D6MAPK1CYP2C19
SCHEMBL9404322 0.85 POLB (0.41) HRH4CYP1A2CYP3A4CYP2D6MAPK1
SCHEMBL9429950 0.83 SMN1; SMN2 (0.54) HRH4HTR3BHTR3ASMN1; SMN2MEN1
SCHEMBL5320912 0.74 HTR3B (0.69) HRH4CYP1A2CYP3A4CYP2D6MAPK1
SCHEMBL3668991 0.73 RXFP1 (0.38) CYP1A2CYP2D6CYP2C19MEN1KMT2A
SCHEMBL30615144 0.73 RXFP1 (0.38) CYP1A2CYP2D6CYP2C19MEN1KMT2A
Hydrochloric Acid SCHEMBL11740107 0.72 HTR3B (0.68) HRH4CYP1A2CYP3A4CYP2D6MAPK1
SCHEMBL8210872 0.72 ELANE (0.76) CNR2
SCHEMBL4090855 0.71 ABCB1 (0.62) CYP1A2CYP3A4CYP2D6MAPK1CYP2C19
SCHEMBL21448035 0.70 DRD2 (0.51) HRH4CYP1A2CYP3A4CYP2D6MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5371080-A Central nervous system disorders NOVO NORDISK A/S 1994-12-06 US disclosed
EP-0619820-A1 IMIDAZOQUINAZOLINE COMPOUNDS AND THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1994-10-19 EP disclosed
WO-1993013103-A1 IMIDAZOQUINAZOLINE COMPOUNDS AND THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1993-07-08 WO disclosed