SCHEMBL9404644

SCHEMBL9404644

O=c1[nH]c2sc3ccc(Cl)cc3c2[nH]c1=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 10/20 0.47
PIM2 Q9P1W9 8/20 0.47
KDM4E B2RXH2 3/20 0.46
CMA1 P23946 1/20 0.45
GRIN2D O15399 2/20 0.42
GRIN3B O60391 2/20 0.42
GRIN1 Q05586 2/20 0.42
GRIN2A Q12879 2/20 0.42
GRIN2B Q13224 2/20 0.42
GRIN2C Q14957 2/20 0.42
GRIN3A Q8TCU5 2/20 0.42
PARP1 P09874 1/20 0.41
ALDH1A1 P00352 2/20 0.38
GAA P10253 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
HPGD P15428 1/20 0.38
PSMB8 P28062 1/20 0.38
CYP2C19 P33261 1/20 0.38
IDO1 P14902 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9404623 0.87 GRIN2D (0.42) PIM1PIM2KDM4ECMA1GRIN2D
SCHEMBL9404641 0.81 PARP1 (0.44) PIM1PIM2PARP1ALDH1A1HPGD
SCHEMBL9404646 0.80 PARP1 (0.36) PARP1
SCHEMBL9404620 0.80 KDM4E (0.42) KDM4EPARP1ALDH1A1GAALMNA
Hydrochloric Acid SCHEMBL9404635 0.80 PARP1 (0.42) PIM1PIM2PARP1ALDH1A1HPGD
SCHEMBL9404642 0.80 PIM1 (0.41) PIM1PIM2HPGDLMNA
SCHEMBL9404640 0.76 PIM1 (0.44) PIM1PIM2KDM4EPARP1HSD17B10
SCHEMBL1908070 0.75 MAPT (0.46) PIM1PIM2KDM4EGRIN2DGRIN3B
SCHEMBL22006353 0.74 PIM1 (0.55) PIM1PIM2KDM4ECMA1
SCHEMBL9404622 0.73 GRIN2D (0.47) PIM1PIM2KDM4EGRIN2DGRIN3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0526588-B1 HETEROCYCLIC COMPOUNDS AND THEIR PREPARATION AND USE NOVO NORDISK AS (DK) 1994-03-09 EP claimed
EP-0526588-B1 HETEROCYCLIC COMPOUNDS AND THEIR PREPARATION AND USE NOVO NORDISK AS (DK) 1994-03-09 EP disclosed
EP-0526588-A1 HETEROCYCLIC COMPOUNDS AND THEIR PREPARATION AND USE. NOVO NORDISK AS (DK) 1993-02-10 EP disclosed
US-5182279-A Antiepileptic, anticonvulsant, anxiolytic, antiischemic NOVO NORDISK A/S (DK) 1993-01-26 US disclosed
WO-1991016325-A1 HETEROCYCLIC COMPOUNDS AND THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1991-10-31 WO disclosed