SCHEMBL9404641

SCHEMBL9404641

Nc1ccc2sc3[nH]c(=O)c(=O)[nH]c3c2c1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 5/20 0.44
MAPT P10636 2/20 0.37
RAB9A P51151 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37
TYMS P04818 2/20 0.36
CA12 O43570 1/20 0.35
CA9 Q16790 1/20 0.35
NPC1 O15118 1/20 0.34
GFER P55789 1/20 0.34
AR P10275 1/20 0.34
NGFR P08138 1/20 0.34
PIM1 P11309 1/20 0.34
PIM2 Q9P1W9 1/20 0.34
NOX4 Q9NPH5 1/20 0.33
PDE10A Q9Y233 1/20 0.32
DAO P14920 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9404635 0.98 PARP1 (0.42) PARP1MAPTRAB9ASMN1; SMN2ALDH1A1
SCHEMBL9404642 0.81 PIM1 (0.41) HPGDTYMSARPIM1PIM2
SCHEMBL9404646 0.81 PARP1 (0.36) PARP1TYMSDAO
SCHEMBL9404644 0.81 PIM1 (0.47) PARP1ALDH1A1HPGDPIM1PIM2
SCHEMBL9404620 0.81 KDM4E (0.42) PARP1MAPTALDH1A1TYMSAR
SCHEMBL9404640 0.78 PIM1 (0.44) PARP1MAPTPIM1PIM2
SCHEMBL1908070 0.77 MAPT (0.46) PARP1MAPTRAB9ASMN1; SMN2ALDH1A1
SCHEMBL11543811 0.75 PARP1 (0.50) PARP1MAPTRAB9ASMN1; SMN2ALDH1A1
SCHEMBL8664533 0.71 RAB9A (0.52) PARP1MAPTRAB9ASMN1; SMN2ALDH1A1
SCHEMBL9404623 0.71 GRIN2D (0.42) PARP1MAPTSMN1; SMN2ALDH1A1GFER

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0526588-B1 HETEROCYCLIC COMPOUNDS AND THEIR PREPARATION AND USE NOVO NORDISK AS (DK) 1994-03-09 EP disclosed
EP-0526588-A1 HETEROCYCLIC COMPOUNDS AND THEIR PREPARATION AND USE. NOVO NORDISK AS (DK) 1993-02-10 EP disclosed
US-5182279-A Antiepileptic, anticonvulsant, anxiolytic, antiischemic NOVO NORDISK A/S (DK) 1993-01-26 US disclosed
WO-1991016325-A1 HETEROCYCLIC COMPOUNDS AND THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1991-10-31 WO disclosed