SCHEMBL9404646

SCHEMBL9404646

O=c1[nH]c2sc3ccc(I)cc3c2[nH]c1=O

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.36
TYMS P04818 2/20 0.34
TUBB4A P04350 1/20 0.32
TUBB P07437 1/20 0.32
TUBA3C P0DPH7 1/20 0.32
TUBA1B P68363 1/20 0.32
TUBA4A P68366 1/20 0.32
TUBB4B P68371 1/20 0.32
TUBB3 Q13509 1/20 0.32
TUBB2A Q13885 1/20 0.32
TUBB8 Q3ZCM7 1/20 0.32
TUBA3E Q6PEY2 1/20 0.32
TUBA1A Q71U36 1/20 0.32
TUBA1C Q9BQE3 1/20 0.32
TUBB6 Q9BUF5 1/20 0.32
TUBB2B Q9BVA1 1/20 0.32
TUBB1 Q9H4B7 1/20 0.32
DAO P14920 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9404641 0.81 PARP1 (0.44) PARP1TYMSDAO
SCHEMBL9404642 0.80 PIM1 (0.41) TYMS
SCHEMBL9404644 0.80 PIM1 (0.47) PARP1
SCHEMBL9404620 0.80 KDM4E (0.42) PARP1TYMSDAO
Hydrochloric Acid SCHEMBL9404635 0.80 PARP1 (0.42) PARP1TYMSDAO
SCHEMBL9404640 0.76 PIM1 (0.44) PARP1
SCHEMBL1908070 0.75 MAPT (0.46) PARP1
SCHEMBL11538149 0.74 CMA1 (0.41) PARP1TYMSTUBB4ATUBBTUBA3C
SCHEMBL9404623 0.70 GRIN2D (0.42) PARP1DAO
Water SCHEMBL9404604 0.69 ALDH1A1 (0.47) PARP1DAO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0526588-B1 HETEROCYCLIC COMPOUNDS AND THEIR PREPARATION AND USE NOVO NORDISK AS (DK) 1994-03-09 EP disclosed
EP-0526588-A1 HETEROCYCLIC COMPOUNDS AND THEIR PREPARATION AND USE. NOVO NORDISK AS (DK) 1993-02-10 EP disclosed
US-5182279-A Antiepileptic, anticonvulsant, anxiolytic, antiischemic NOVO NORDISK A/S (DK) 1993-01-26 US disclosed
WO-1991016325-A1 HETEROCYCLIC COMPOUNDS AND THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1991-10-31 WO disclosed