SCHEMBL9406263

SCHEMBL9406263

CCCCC[C@H]1CC[C@H](CCc2cccc(F)c2F)CC1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.40
MAOB P27338 1/20 0.40
RIPK1 Q13546 1/20 0.38
BCHE P06276 1/20 0.36
GRM2 Q14416 1/20 0.34
P2RX7 Q99572 1/20 0.34
DRD2 P14416 1/20 0.34
DRD3 P35462 1/20 0.34
HTR2A P28223 3/20 0.33
HTR2C P28335 3/20 0.33
OPRM1 P35372 1/20 0.33
SIGMAR1 Q99720 1/20 0.33
CYP1A2 P05177 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
APLNR P35414 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9406269 1.00 MAOA (0.40) MAOAMAOBRIPK1BCHEGRM2
SCHEMBL8983091 0.96 MAOA (0.38) MAOAMAOBRIPK1BCHEGRM2
SCHEMBL8983100 0.96 MAOA (0.38) MAOAMAOBRIPK1BCHEGRM2
SCHEMBL17527894 0.89 MAOA (0.43) MAOAMAOBRIPK1P2RX7HTR2A
SCHEMBL8375636 0.88 MAOA (0.51) MAOAMAOBBCHEGRM2HTR2A
SCHEMBL9251813 0.87 CYP1A2 (0.34) MAOAMAOBRIPK1P2RX7HTR2A
SCHEMBL9251807 0.87 CYP1A2 (0.34) MAOAMAOBRIPK1P2RX7HTR2A
SCHEMBL10708324 0.86 CYP1A2 (0.38) MAOAMAOBHTR2AHTR2CCYP1A2
SCHEMBL10708319 0.86 CYP1A2 (0.38) MAOAMAOBHTR2AHTR2CCYP1A2
SCHEMBL4801585 0.85 MAOA (0.40) MAOAMAOBRIPK1P2RX7HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0363458-B1 2,3-DIFLUOROBENZENES MERCK PATENT GMBH (DE) 1994-08-03 EP disclosed
US-5279764-A Dihalogenobenzene derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1994-01-18 US disclosed
US-5211878-A Difluorobenzonitrile derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1993-05-18 US disclosed
EP-0364538-B1 DIFLUOROBENZOL DERIVATIVES MERCK PATENT GmbH (DE) 1992-05-06 EP disclosed
US-5087764-A Deprotonation of a 1-substituted-2,3-difluorobenzene using an organometallic compound and reacting the reaction product with an electrophile Merck Patent Gesellschaft mit beschrankter Hafung (DE) 1992-02-11 US disclosed
EP-0364538-A1 DIFLUOROBENZOL DERIVATIVES. MERCK PATENT GMBH (DE) 1990-04-25 EP disclosed
EP-0363458-A1 2,3-DIFLUOROBENZENES. MERCK PATENT GMBH (DE) 1990-04-18 EP disclosed
WO-1989008629-A1 PROCESS FOR PREPARING 2,3-DIFLUOROBENZENES MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1989-09-21 WO disclosed
WO-1989008633-A1 DIFLUOROBENZOL DERIVATIVES MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1989-09-21 WO disclosed