SCHEMBL9407965

SCHEMBL9407965

O=C(O)[C@H]1CC[C@H](c2nnc(-c3ccc(N4CCN(Cc5ccccc5)CC4)cc3)s2)CC1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.55
HTR2C P28335 1/20 0.55
HTR2B P41595 1/20 0.55
DRD4 P21917 3/20 0.46
TSHR P16473 1/20 0.46
USP2 O75604 3/20 0.45
ALDH1A1 P00352 2/20 0.45
MAPT P10636 3/20 0.44
HTT P42858 1/20 0.44
ATM Q13315 1/20 0.44
ESR1 P03372 1/20 0.44
ESR2 Q92731 1/20 0.44
S1PR1 P21453 2/20 0.44
S1PR3 Q99500 1/20 0.44
HTR7 P34969 2/20 0.43
MAPK1 P28482 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
HDAC3 O15379 1/20 0.41
HDAC4 P56524 1/20 0.41
HDAC1 Q13547 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9407966 1.00 HTR2A (0.55) HTR2AHTR2CHTR2BDRD4TSHR
SCHEMBL9408081 0.88 ALDH1A1 (0.55) HTR2AHTR2CHTR2BUSP2ALDH1A1
SCHEMBL9408089 0.88 ALDH1A1 (0.55) HTR2AHTR2CHTR2BUSP2ALDH1A1
SCHEMBL9407953 0.82 TSHR (0.40) TSHRUSP2ALDH1A1MAPT
SCHEMBL9407948 0.82 TSHR (0.40) TSHRUSP2ALDH1A1MAPT
Hydrochloric Acid SCHEMBL9407957 0.81 TSHR (0.39) TSHRUSP2ALDH1A1MAPT
SCHEMBL13098786 0.78 MAPT (0.38) TSHRUSP2ALDH1A1MAPTS1PR1
SCHEMBL29987937 0.77 CSNK2A2 (0.44) ALDH1A1MAPTHTTSMN1; SMN2HDAC3
SCHEMBL13098918 0.74 MAPT (0.35) USP2ALDH1A1MAPTS1PR1MAPK1
SCHEMBL13099111 0.74 USP2 (0.41) TSHRUSP2ALDH1A1MAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0608858-A1 5-Membered heterocycles as aggregation inhibitors Dr. Karl Thomae GmbH (DE) 1994-08-03 EP disclosed