SCHEMBL9407948

SCHEMBL9407948

O=C(O)[C@H]1CC[C@H](c2nnc(-c3ccc(N4CCNCC4)cc3)s2)CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.40
USP2 O75604 2/20 0.40
ALDH1A1 P00352 2/20 0.40
HSD17B10 Q99714 1/20 0.40
MAPKAPK2 P49137 4/20 0.39
CSNK2A2 P19784 1/20 0.38
CSNK2A1 P68400 1/20 0.38
ABL1 P00519 1/20 0.38
TNKS O95271 1/20 0.37
PARP1 P09874 1/20 0.37
PARP2 Q9UGN5 1/20 0.37
ACVR1 Q04771 2/20 0.36
AKR1C3 P42330 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
ITGA2B P08514 1/20 0.36
USP28 Q96RU2 1/20 0.35
USP25 Q9UHP3 1/20 0.35
HTR3E A5X5Y0 1/20 0.35
HTR3B O95264 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9407953 1.00 TSHR (0.40) TSHRUSP2ALDH1A1HSD17B10MAPKAPK2
Hydrochloric Acid SCHEMBL9407957 0.99 TSHR (0.39) TSHRUSP2ALDH1A1HSD17B10MAPKAPK2
SCHEMBL13099208 0.87 MAPT (0.42) USP2MAPKAPK2ABL1ACVR1USP28
Hydrochloric Acid SCHEMBL9408126 0.86 MAPT (0.41) USP2MAPKAPK2ABL1ACVR1USP28
Hydrochloric Acid SCHEMBL9408037 0.84 LGMN (0.45) ALDH1A1ACVR1NPC1USP28USP25
SCHEMBL9244763 0.83 NPC1 (0.50) TSHRCSNK2A2CSNK2A1PARP1PARP2
SCHEMBL9244757 0.83 NPC1 (0.50) TSHRCSNK2A2CSNK2A1PARP1PARP2
SCHEMBL9407966 0.82 HTR2A (0.55) TSHRUSP2ALDH1A1MAPT
SCHEMBL9407965 0.82 HTR2A (0.55) TSHRUSP2ALDH1A1MAPT
SCHEMBL13098786 0.82 MAPT (0.38) TSHRUSP2ALDH1A1CSNK2A2CSNK2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0608858-A1 5-Membered heterocycles as aggregation inhibitors Dr. Karl Thomae GmbH (DE) 1994-08-03 EP disclosed