Trifluomeprazine

Trifluomeprazine

SCHEMBL941053

CC(CN(C)C)CN1c2ccccc2Sc2ccc(C(F)(F)F)cc21

nearest known ligand 0.72

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 5/20 0.72
ADRA2A P08913 5/20 0.72
CHRM1 P11229 5/20 0.72
DRD1 P21728 5/20 0.72
ADRA1A P35348 5/20 0.72
DRD3 P35462 5/20 0.72
KCNH2 Q12809 5/20 0.72
CHRM2 P08172 4/20 0.72
TBXA2R P21731 4/20 0.72
OPRM1 P35372 4/20 0.72
SLC6A2 P23975 4/20 0.72
SLC6A4 P31645 4/20 0.72
SLC6A3 Q01959 4/20 0.72
ABCB11 O95342 2/20 0.72
HRH3 Q9Y5N1 2/20 0.72
CYP2D6 P10635 5/20 0.68
LMNA P02545 5/20 0.67
MAPK1 P28482 4/20 0.67
CYP3A4 P08684 4/20 0.67
CYP1A2 P05177 3/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Triflupromazine SCHEMBL5311245 0.92 CYP2D6 (0.80) HTR1AADRA2ACHRM1DRD1ADRA1A
SCHEMBL26000537 0.87 FPR2 (0.75) HTR1AADRA2ACHRM1DRD1ADRA1A
SCHEMBL2892321 0.86 CYP2D6 (0.71) HTR1AADRA2ACHRM1DRD1ADRA1A
SCHEMBL2892325 0.86 CYP2D6 (0.71) HTR1AADRA2ACHRM1DRD1ADRA1A
Triflupromazine SCHEMBL20610220 0.85 CYP2D6 (0.71) HTR1AADRA2ACHRM1DRD1ADRA1A
Methylpromazine SCHEMBL18993 0.85 CHRM2 (1.00) HTR1AADRA2ACHRM1DRD1ADRA1A
Methylpromazine SCHEMBL18994 0.85 CHRM2 (1.00) HTR1AADRA2ACHRM1DRD1ADRA1A
Methylpromazine SCHEMBL29354434 0.85 CHRM2 (1.00) HTR1AADRA2ACHRM1DRD1ADRA1A
Triflupromazine SCHEMBL13724400 0.85 CYP2D6 (0.68) HTR1AADRA2ACHRM1DRD1ADRA1A
SCHEMBL13284571 0.84 CHRM2 (0.78) HTR1AADRA2ACHRM1DRD1ADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 160 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102935068-B Preparation method of liposome entrapping water-soluble medicines ZHEJIANG HISUN PHARM CO LTD 2014-12-17 CN claimed
CN-102935068-A Preparation method of liposome entrapping water-soluble medicines ZHEJIANG HISUN PHARM CO LTD 2013-02-20 CN claimed
CN-101426495-A CB1 antagonists and inverse agonists AMPLA PHARMACEUTICALS INC (US) 2009-05-06 CN claimed
WO-2025093589-A1 HETEROARYL AMIDE DERIVATIVES AS SODIUM CHANNEL INHIBITORS CHIESI FARMACEUTICI S.P.A. (IT) 2025-05-08 WO disclosed
WO-2025093590-A1 HETEROARYL ESTER DERIVATIVES AS SODIUM CHANNEL INHIBITORS CHIESI FARMACEUTICI S.P.A. (IT) 2025-05-08 WO disclosed
WO-2024189607-A1 METHODS AND BIOAVAILABLE HIGHLY PERMEABLE COMPOUNDS FOR DISEASES TREATMENT DIDENKO KIRILL (MX) 2024-09-19 WO disclosed
WO-2023037254-A1 METHODS AND COMPOUNDS FOR TREATING CORONAVIRIDAE VIRUS INFECTIONS DIDENKO KIRILL (MX) 2023-03-16 WO disclosed
US-10376522-B2 Triarylmethane analogs and their use in treating cancers EMORY UNIVERSITY (US) 2019-08-13 US disclosed
US-9586899-B2 Synthetic process for aminocyclohexyl ether compounds CARDIOME PHARMA CORP. (CA) 2017-03-07 US disclosed
US-20170000801-A1 TRIARYLMETHANE ANALOGS AND THEIR USE IN TREATING CANCERS THE US GOVERNMENT AS REPRESENTED BY THE DEPARTMENT OF VETERAN AFFAIRS 2017-01-05 US disclosed
US-20170000801-A1 TRIARYLMETHANE ANALOGS AND THEIR USE IN TREATING CANCERS THE US GOVERNMENT AS REPRESENTED BY THE DEPARTMENT OF VETERAN AFFAIRS 2017-01-05 US disclosed
US-20020102215-A1 Diagnostic/therapeutic agents NYCOMED IMAGING AS 2002-08-01 US disclosed
US-20020040359-A1 Method and apparatus for normalizing and converting structured content ORACLE INTERNATIONAL CORPORATION 2002-04-04 US disclosed
US-20020040359-A1 Method and apparatus for normalizing and converting structured content ORACLE INTERNATIONAL CORPORATION 2002-04-04 US disclosed
WO-2002001401-A1 METHOD AND APPARATUS FOR NORMALIZING AND CONVERTING STRUCTURED CONTENT ONEREALM INC. (US) 2002-01-03 WO disclosed
WO-2002001401-A1 METHOD AND APPARATUS FOR NORMALIZING AND CONVERTING STRUCTURED CONTENT ONEREALM INC. (US) 2002-01-03 WO disclosed
WO-2001096335-A1 IMIDAZO[1,2-A]PYRIDINE ETHER COMPOUNDS AS ION CHANNEL MODULATORS CARDIOME PHARMA CORP. (CA) 2001-12-20 WO disclosed
US-6331289-B1 ULTRASOUND CONTRAST AGENTS, SUSPENSION IN AQUEOUS CARRIER LIQUID OF A REPORTER COMPRISING GAS-CONTAINING OR GAS-GENERATING MATERIAL, AGENT CAPABLE OF FORMING AT LEAST TWO TYPES OF BINDING PAIRS WITH TARGET; REPORTER BEING CONJUGATED NYCOMED IMAGING AS (NO) 2001-12-18 US disclosed
US-6264917-B1 MIXTURE OF GAS FILLED MICROBUBBLES AND RELEASING AGENT NYCOMED IMAGING AS (NO) 2001-07-24 US disclosed
US-6261537-B1 TARGETS AND ULTRASOUND DIAGNOSIS OF ACTIVE MATERIALS, AQUEOUS CARRIER LIQUIDS, CARRIERS AND FILM FORMING SURFACTANT PHOSPHATIDES NYCOMED IMAGING AS (NO) 2001-07-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170000801-A1 TRIARYLMETHANE ANALOGS AND THEIR USE IN TREATING CANCERS TK2, TXNRD2, TXN2 HTR1A 3040/4885ADRA2A 2595/4885CHRM1 4646/4885
US-10376522-B2 Triarylmethane analogs and their use in treating cancers TK2, TXNRD2, TXN2 HTR1A 3045/4885ADRA2A 2553/4885CHRM1 4644/4885
US-20020102215-A1 Diagnostic/therapeutic agents BID, FUS, FABP1 HTR1A 4030/4885ADRA2A 2412/4885CHRM1 4583/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.