SCHEMBL9412262

SCHEMBL9412262

O=C1CCc2cc(N3CCN(Cc4ccc(Cl)cc4)CC3)ccc2N1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 7/20 0.60
DRD2 P14416 5/20 0.60
DRD3 P35462 4/20 0.60
HTR1A P08908 2/20 0.60
CHRM5 P08912 1/20 0.60
ADRA2A P08913 1/20 0.60
ADRA2B P18089 1/20 0.60
HTR2A P28223 1/20 0.60
ADRA1B P35368 1/20 0.60
TMEM97 Q5BJF2 1/20 0.60
SIGMAR1 Q99720 1/20 0.60
KCNH2 Q12809 2/20 0.58
MAPT P10636 2/20 0.51
SLC6A4 P31645 3/20 0.50
SLC6A2 P23975 2/20 0.50
SLC6A3 Q01959 2/20 0.50
KDM4E B2RXH2 2/20 0.48
ALDH1A1 P00352 2/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
NR3C1 P04150 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11194558 0.89 DRD4 (0.59) DRD4DRD2DRD3HTR1ACHRM5
SCHEMBL11196367 0.89 SLC6A4 (0.52) DRD4DRD2DRD3HTR1ACHRM5
Hydrochloric Acid SCHEMBL9412123 0.88 DRD4 (0.58) DRD4DRD2DRD3HTR1ACHRM5
SCHEMBL9412142 0.86 DRD4 (0.61) DRD4DRD2DRD3HTR1AKCNH2
SCHEMBL23765267 0.84 DRD4 (0.49) DRD4DRD2DRD3HTR1ACHRM5
SCHEMBL11197642 0.82 ALDH1A1 (0.69) DRD4DRD2DRD3HTR1ACHRM5
SCHEMBL9412170 0.80 KCNH2 (0.69) KCNH2SLC6A4ALDH1A1SMN1; SMN2NR3C1
SCHEMBL10837507 0.80 KCNH2 (0.55) DRD4DRD2DRD3HTR1ACHRM5
SCHEMBL10837503 0.80 KCNH2 (0.55) DRD4DRD2DRD3HTR1ACHRM5
SCHEMBL16035044 0.80 KCNH2 (0.55) DRD4DRD2DRD3HTR1ACHRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0623598-A1 APOPTOSIS REGULATOR OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-11-09 EP disclosed
US-4415572-A CARDIOTONIC AND INOTROPIC AGENTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1983-11-15 US disclosed