SCHEMBL9412461

SCHEMBL9412461

Cn1c(-c2ccc(C#N)cc2)nc2c1c(=O)[nH]c(=O)n2C

nearest known ligand 0.68

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.59
ALDH1A1 P00352 6/20 0.59
HPGD P15428 3/20 0.59
PKM P14618 1/20 0.53
MAPT P10636 2/20 0.52
HSD17B10 Q99714 2/20 0.52
UBE2N P61088 1/20 0.52
NPSR1 Q6W5P4 2/20 0.46
TSHR P16473 2/20 0.45
GAA P10253 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
CYP3A4 P08684 1/20 0.42
MAPK1 P28482 1/20 0.42
PMP22 Q01453 1/20 0.42
ADORA2A P29274 1/20 0.42
ADORA2B P29275 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7057695 0.81 KDM4E (0.62) KDM4EALDH1A1HPGDPKMMAPT
SCHEMBL9412635 0.80 KDM4E (0.46) KDM4EALDH1A1HPGDPKMMAPT
SCHEMBL25090486 0.80 ADORA2B (0.68) KDM4EALDH1A1HPGDADORA2AADORA2B
SCHEMBL5437075 0.74 KDM4E (0.41) KDM4EALDH1A1HPGDPKMMAPT
SCHEMBL5449103 0.74 KDM4E (0.41) KDM4EALDH1A1HPGDPKMMAPT
SCHEMBL6876786 0.71 GAA (0.58) KDM4EALDH1A1HPGDHSD17B10NPSR1
SCHEMBL5642013 0.70 MEN1 (0.55) ALDH1A1MAPTNPSR1TSHRMAPK1
SCHEMBL9287667 0.70 KDM4E (0.38) KDM4EALDH1A1HPGDPKMMAPT
SCHEMBL16598824 0.68 SMN1; SMN2 (0.47) KDM4EALDH1A1MAPTHSD17B10TSHR
SCHEMBL18865648 0.67 CYP11B2 (0.45) ALDH1A1MAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0611660-A2 Condensed 5-membered heterocycles, process for their preparation and medicines containing these compounds Dr. Karl Thomae GmbH (DE) 1994-08-24 EP disclosed