SCHEMBL9416249

SCHEMBL9416249

COc1ccc(C(=S)SC(=O)CO)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.48
CES1 P23141 1/20 0.48
PLK1 P53350 1/20 0.47
CA1 P00915 5/20 0.47
CA2 P00918 5/20 0.47
HDAC3 O15379 6/20 0.47
HDAC4 P56524 6/20 0.47
HDAC1 Q13547 6/20 0.47
HDAC7 Q8WUI4 6/20 0.47
HDAC2 Q92769 6/20 0.47
HDAC10 Q969S8 6/20 0.47
HDAC11 Q96DB2 6/20 0.47
HDAC8 Q9BY41 6/20 0.47
HDAC6 Q9UBN7 6/20 0.47
HDAC9 Q9UKV0 6/20 0.47
HDAC5 Q9UQL6 6/20 0.47
GSK3B P49841 1/20 0.46
PARP1 P09874 1/20 0.46
PARP10 Q53GL7 1/20 0.46
PARP2 Q9UGN5 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9547489 0.81 CES2 (0.53) CES2CES1PLK1CA1CA2
SCHEMBL2705457 0.81 HDAC1 (0.44) CES2CES1HDAC3HDAC4HDAC1
SCHEMBL828942 0.77 HDAC3 (0.44) CES2CES1HDAC3HDAC4HDAC1
SCHEMBL9416245 0.77 RAB9A (0.47) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL237978 0.74 CES2 (0.52) CES2CES1CA1CA2PARP1
SCHEMBL9416228 0.73 CES2 (0.48) CES2CES1HDAC1HDAC8GSK3B
SCHEMBL9416250 0.73 MAPT (0.67) CES2CES1CA1CA2HDAC3
SCHEMBL5192809 0.72 NPC1 (0.50) CES2CES1CA1CA2PARP1
SCHEMBL505810 0.72 HDAC3 (0.68) CES2CES1CA1CA2HDAC3
SCHEMBL10908525 0.72 HDAC3 (0.59) CES2CES1HDAC3HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0601520-A1 Trifluorothymidine derivatives, process for producing the same and anti-cancer agent containing the same MITSUI TOATSU CHEMICALS, Inc. (JP) 1994-06-15 EP disclosed