SCHEMBL9418949

SCHEMBL9418949

CC1(C)CC(=O)CCc2ccc(Br)cc21

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CMA1 P23946 1/20 0.42
AHR P35869 1/20 0.42
TDP2 O95551 2/20 0.40
TDP1 Q9NUW8 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
KDM1A O60341 1/20 0.39
BRD4 O60885 1/20 0.38
SRD5A1 P18405 1/20 0.37
PARP1 P09874 1/20 0.37
PARP10 Q53GL7 1/20 0.37
BACE1 P56817 5/20 0.35
APP P05067 1/20 0.35
PDE4B Q07343 1/20 0.35
TYMS P04818 1/20 0.35
METAP1 P53582 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HSD17B3 P37058 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9419023 0.88 TDP2 (0.42) CMA1AHRTDP2TDP1L3MBTL1
SCHEMBL7796330 0.84 CMA1 (0.47) CMA1AHRTDP2TDP1L3MBTL1
SCHEMBL9418964 0.80 CMA1 (0.42) CMA1AHRTDP2L3MBTL1BRD4
SCHEMBL8370875 0.76 TDP2 (0.47) CMA1AHRTDP2TDP1L3MBTL1
SCHEMBL1706762 0.76 KDM1A (0.53) CMA1AHRTDP2TDP1L3MBTL1
SCHEMBL29804270 0.76 KDM1A (0.53) CMA1AHRTDP2TDP1L3MBTL1
SCHEMBL2012588 0.73 BACE1 (0.51) CMA1AHRKDM1ABACE1APP
SCHEMBL3361527 0.71 PGR (0.55) CMA1AHRTDP2PDE4BMETAP1
SCHEMBL6674280 0.71 BACE1 (0.47) KDM1ABACE1APP
SCHEMBL10182282 0.71 TDP1 (0.48) CMA1AHRTDP2TDP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0315071-B1 Benzocyclohepten derivatives, their preparation and utilisation for pharmaceutics HOFFMANN LA ROCHE (CH) 1994-07-20 EP disclosed
US-4992574-A Skin disorders, antiallergens, antiinflammatory agent HOFFMANN-LA ROCHE INC. (US) 1991-02-12 US disclosed
EP-0315071-A2 Benzocyclohepten derivatives, their preparation and utilisation for pharmaceutics F. HOFFMANN-LA ROCHE AG (CH) 1989-05-10 EP disclosed