SCHEMBL9419974

SCHEMBL9419974

Cc1cc(Cl)c(Cl)c(C)c1Cl

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 5/20 0.43
CHRM1 P11229 1/20 0.43
ALOX15 P16050 1/20 0.43
MAOA P21397 1/20 0.43
TBXA2R P21731 1/20 0.43
ADRA1A P35348 1/20 0.43
HTR2B P41595 1/20 0.43
SIRT1 Q96EB6 1/20 0.43
ALDH1A1 P00352 3/20 0.43
GAA P10253 1/20 0.43
MAPT P10636 1/20 0.43
RAPGEF4 Q8WZA2 4/20 0.41
CD44 P16070 1/20 0.36
HPGD P15428 5/20 0.35
HSD17B10 Q99714 5/20 0.35
TSHR P16473 4/20 0.35
CRHBP P24387 1/20 0.35
CRHR2 Q13324 1/20 0.35
CASP1 P29466 1/20 0.35
HSP90AA1 P07900 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1003476 0.84 CYP3A4 (0.50) CYP3A4CHRM1ALOX15MAOATBXA2R
SCHEMBL1547849 0.84 CYP3A4 (0.56) CYP3A4CHRM1ALOX15MAOATBXA2R
SCHEMBL10913798 0.82 CYP3A4 (0.40) CYP3A4CHRM1ALOX15MAOATBXA2R
SCHEMBL31120437 0.82 CYP3A4 (0.40) CYP3A4CHRM1ALOX15MAOATBXA2R
SCHEMBL1019625 0.82 CYP3A4 (0.43) CYP3A4CHRM1ALOX15MAOATBXA2R
SCHEMBL31497683 0.82 CYP3A4 (0.43) CYP3A4CHRM1ALOX15MAOATBXA2R
SCHEMBL29380985 0.81 CYP3A4 (0.48) CYP3A4CHRM1ALOX15MAOATBXA2R
SCHEMBL31519176 0.79 CYP3A4 (0.59) CYP3A4CHRM1ALOX15MAOATBXA2R
SCHEMBL2260986 0.79 CYP3A4 (0.59) CYP3A4CHRM1ALOX15MAOATBXA2R
SCHEMBL1006177 0.77 CYP3A4 (0.43) CYP3A4CHRM1ALOX15MAOATBXA2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0563033-A4 PROCESS FOR PREPARING 3-TRIFLUOROMETHYL BENZYL CHLORIDE CHEVRON RES & TECH (US) 1994-05-18 EP claimed
EP-0563033-A1 PROCESS FOR PREPARING 3-TRIFLUOROMETHYL BENZYL CHLORIDE. CHEVRON RES & TECH (US) 1993-10-06 EP claimed
WO-1992007820-A1 PROCESS FOR PREPARING 3-TRIFLUOROMETHYL BENZYL CHLORIDE CHEVRON RESEARCH AND TECHNOLOGY COMPANY (US) 1992-05-14 WO claimed
US-4059610-A Process for preparing isocyanic acid derivatives KAO SOAP CO., LTD. (JA) 1977-11-22 US claimed
US-20170267717-A1 Novel method for the production of 18F-labeled active esters and their application exemplified by the preparation of a PSMA-specific PET-tracer MAX-PLANCK-GESELLSCHAFT ZUR FOERDERUNG DER WISSENSCHAFTEN E.V. (DE) 2017-09-21 US disclosed
EP-0563033-A4 PROCESS FOR PREPARING 3-TRIFLUOROMETHYL BENZYL CHLORIDE CHEVRON RES & TECH (US) 1994-05-18 EP disclosed
EP-0563033-A1 PROCESS FOR PREPARING 3-TRIFLUOROMETHYL BENZYL CHLORIDE. CHEVRON RES & TECH (US) 1993-10-06 EP disclosed
WO-1992007820-A1 PROCESS FOR PREPARING 3-TRIFLUOROMETHYL BENZYL CHLORIDE CHEVRON RESEARCH AND TECHNOLOGY COMPANY (US) 1992-05-14 WO disclosed
US-4059610-A Process for preparing isocyanic acid derivatives KAO SOAP CO., LTD. (JA) 1977-11-22 US disclosed
US-4056547-A FROM AN ALKALI METAL OR AMMONIUM CYANATE AND A BENZYL CHLORIDE, CATALYST KAO SOAP CO., LTD. (JA) 1977-11-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170267717-A1 Novel method for the production of 18F-labeled active esters and their application exemplified by the preparation of a PSMA-specific PET-tracer FGB, F13B, FAP CYP3A4 1540/4885CHRM1 3864/4885ALOX15 3406/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.