SCHEMBL9422178

SCHEMBL9422178

Oc1nc2ccc(-c3ccc4nc(O)c(O)nc4c3)cc2nc1O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRC P12931 2/20 0.43
KDM4E B2RXH2 3/20 0.40
PIK3R1 P27986 2/20 0.39
PIK3CA P42336 2/20 0.39
NPC1 O15118 1/20 0.38
POLB P06746 1/20 0.38
RAB9A P51151 1/20 0.38
CYP2C19 P33261 1/20 0.38
ESR1 P03372 3/20 0.38
ESR2 Q92731 3/20 0.38
APP P05067 1/20 0.38
MAP4K4 O95819 1/20 0.37
CDK8 P49336 1/20 0.37
CLK2 P49760 1/20 0.37
CDK7 P50613 1/20 0.37
CDK9 P50750 1/20 0.37
CDK5 Q00535 1/20 0.37
ACVR1 Q04771 1/20 0.37
ROCK1 Q13464 1/20 0.37
DYRK1A Q13627 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14582918 0.79 ALDH1A1 (0.50) KDM4ECYP2C19ESR1ESR2PIK3CG
SCHEMBL11038516 0.77 PIK3R1 (0.41) SRCPIK3R1PIK3CAPOLBRAB9A
SCHEMBL10545679 0.77 KMT2A (0.64) KDM4ENPC1RAB9AESR1ESR2
SCHEMBL9979784 0.76 NQO1 (0.44) KDM4ECYP2C19MAPTNQO2
SCHEMBL7173382 0.76 NQO2 (0.62) SRCKDM4EPIK3R1PIK3CANPC1
SCHEMBL10553377 0.75 NQO2 (0.64) KDM4ENPC1RAB9AMEN1KMT2A
SCHEMBL10851061 0.75 KDM4E (0.69) KDM4ENPC1RAB9ACYP2C19APP
SCHEMBL29581721 0.75 HSD17B10 (0.53) KDM4EPIK3R1PIK3CAPOLBDYRK1A
SCHEMBL6109123 0.75 PABPC1 (0.50) KDM4EPIK3R1PIK3CACYP2C19ALDH1A1
SCHEMBL6109697 0.75 HSD17B10 (0.53) KDM4EPIK3R1PIK3CAPOLBDYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 23 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0231373-B1 A PROCESS FOR THE PRODUCTION OF A LIQUID CRYSTALLINE EXTENDED CHAIN POLYMER COMPOSITION THE DOW CHEMICAL COMPANY (US) 1991-01-30 EP claimed
EP-0119271-B1 LIQUID CRYSTALLINE POLYMER COMPOSITIONS, PROCESS, AND PRODUCTS SRI INTERNATIONAL (US) 1990-07-11 EP claimed
EP-0231373-A4 A PROCESS FOR THE PRODUCTION OF A LIQUID CRYSTALLINE EXTENDED CHAIN POLYMER COMPOSITION. COMMTECH INTERNAT (US) 1988-12-22 EP claimed
US-4772678-A HIGH-MOLECULAR-WEIGHT CHAIN-EXTENDED N-HETEROCYCLIC POLYMERS PREPARED USING A NON-OXIDIZING STRONG ACID AS SOLVENT; HIGH-STRENGTH FIBERS, FILMS, FIBRIDS AND STRUCTURES COMMTECH INTERNATIONAL MANAGEMENT CORPORATION (US) 1988-09-20 US claimed
US-4703103-A POLYPHOSPHORIC ACID CATALYST COMMTECH INTERNATIONAL (US) 1987-10-27 US claimed
EP-0231373-A1 A PROCESS FOR THE PRODUCTION OF A LIQUID CRYSTALLINE EXTENDED CHAIN POLYMER COMPOSITION. COMMTECH INT (US) 1987-08-12 EP claimed
WO-1987000844-A1 A PROCESS FOR THE PRODUCTION OF A LIQUID CRYSTALLINE EXTENDED CHAIN POLYMER COMPOSITION COMMTECH INTERNATIONAL (US) 1987-02-12 WO claimed
WO-1985004178-A1 LIQUID CRYSTALLINE POLYMER COMPOSITIONS, PROCESS, AND PRODUCTS SRI INTERNATIONAL (US) 1985-09-26 WO claimed
US-4533693-A ANISOTROPIC; FIBERS, FILMS SRI INTERNATIONAL (US) 1985-08-06 US claimed
EP-0119271-A4 LIQUID CRYSTALLINE POLYMER COMPOSITIONS, PROCESS, AND PRODUCTS. STANFORD RES INST INT (US) 1985-07-01 EP claimed
EP-0119271-A1 LIQUID CRYSTALLINE POLYMER COMPOSITIONS, PROCESS, AND PRODUCTS. STANFORD RES INST INT (US) 1984-09-26 EP claimed
EP-0119192-A1 LIQUID CRYSTALLINE POLYMER COMPOSITIONS, PROCESS, AND PRODUCTS SRI INTERNATIONAL (US) 1984-09-26 EP claimed
WO-1984001160-A1 LIQUID CRYSTALLINE POLYMER COMPOSITIONS, PROCESS, AND PRODUCTS STANFORD RES INST INT (US) 1984-03-29 WO claimed
WO-1984001162-A1 LIQUID CRYSTALLINE POLYMER COMPOSITIONS, PROCESS, AND PRODUCTS STANFORD RES INST INT (US) 1984-03-29 WO claimed
US-5374706-A High molecular weight ordered polybenzoxazole fibers THE DOW CHEMICAL COMPANY (US) 1994-12-20 US disclosed
EP-0231373-B1 A PROCESS FOR THE PRODUCTION OF A LIQUID CRYSTALLINE EXTENDED CHAIN POLYMER COMPOSITION THE DOW CHEMICAL COMPANY (US) 1991-01-30 EP disclosed
EP-0231373-A4 A PROCESS FOR THE PRODUCTION OF A LIQUID CRYSTALLINE EXTENDED CHAIN POLYMER COMPOSITION. COMMTECH INTERNAT (US) 1988-12-22 EP disclosed
EP-0119271-A4 LIQUID CRYSTALLINE POLYMER COMPOSITIONS, PROCESS, AND PRODUCTS. STANFORD RES INST INT (US) 1985-07-01 EP disclosed
EP-0119271-A1 LIQUID CRYSTALLINE POLYMER COMPOSITIONS, PROCESS, AND PRODUCTS. STANFORD RES INST INT (US) 1984-09-26 EP disclosed
WO-1984001162-A1 LIQUID CRYSTALLINE POLYMER COMPOSITIONS, PROCESS, AND PRODUCTS STANFORD RES INST INT (US) 1984-03-29 WO disclosed