Iodide

Iodide

SCHEMBL9424070

CSC(=N)Nc1c(C)cccc1N1CCCCC1.I

nearest known ligand 0.46

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHECHRM1CHRM3CHRNA1CHRNB1CHRNDCHRNECHRNG

The experimentally established mechanism targets of Iodide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 5/20 0.46
MAPT P10636 5/20 0.46
NPSR1 Q6W5P4 3/20 0.46
POLB P06746 3/20 0.44
ATM Q13315 5/20 0.44
ALDH1A1 P00352 4/20 0.41
KMT2A Q03164 4/20 0.41
LMNA P02545 3/20 0.41
MEN1 O00255 3/20 0.41
MAPK1 P28482 4/20 0.39
USP2 O75604 1/20 0.39
ALOX15 P16050 1/20 0.39
GAA P10253 3/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
TDP1 Q9NUW8 2/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
GFER P55789 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Iodide SCHEMBL9424394 0.86 SCN9A (0.47) L3MBTL1MAPTNPSR1POLBALDH1A1
SCHEMBL9059228 0.83 MAPT (0.48) L3MBTL1MAPTNPSR1POLBATM
Iodide SCHEMBL9424005 0.78 NPSR1 (0.56) L3MBTL1MAPTNPSR1POLBATM
SCHEMBL12004117 0.77 L3MBTL1 (0.47) L3MBTL1MAPTNPSR1POLBATM
SCHEMBL9423957 0.77 L3MBTL1 (0.48) L3MBTL1MAPTNPSR1POLBATM
Iodide SCHEMBL9423985 0.77 L3MBTL1 (0.54) L3MBTL1MAPTNPSR1POLBATM
SCHEMBL9059533 0.76 L3MBTL1 (0.47) L3MBTL1MAPTNPSR1POLBATM
SCHEMBL9060599 0.75 DRD2 (0.48) L3MBTL1MAPTNPSR1POLBATM
Iodide SCHEMBL9060369 0.70 SCN9A (0.47) MAPTNPSR1POLBALDH1A1KMT2A
Iodide SCHEMBL9060364 0.70 SCN9A (0.47) MAPTNPSR1POLBALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5373008-A Phenylamidine and phenylguanidine derivatives and their use as anti-diabetic agents THE BOOTS COMPANT PLC. (GB) 1994-12-13 US disclosed
US-5223498-A Hypoglycemic agents THE BOOTS COMPANY PLC (GB) 1993-06-29 US disclosed
EP-0385038-B1 ORTHO-SUBSTITUTED PHENYL AMIDINE AND PHENYL GUANIDINE DERIVATIVES AND ANTIDIABETIC OR HYPOGLYCAEMIC AGENTS CONTAINING THEM The Boots Company PLC (GB) 1993-06-02 EP disclosed
EP-0385038-A1 Ortho-substituted phenyl amidine and phenyl guanidine derivatives and antidiabetic or hypoglycaemic agents containing them The Boots Company PLC (GB) 1990-09-05 EP disclosed