SCHEMBL9425903

SCHEMBL9425903

CCCCN(C)C(=O)CCc1ccc(OCc2ccccn2)c(OCc2ccccn2)c1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
RAF1 P04049 7/20 0.51
MAP2K1 Q02750 7/20 0.51
HDAC1 Q13547 1/20 0.49
HDAC2 Q92769 1/20 0.49
APP P05067 1/20 0.49
KDM4E B2RXH2 3/20 0.47
ALDH1A1 P00352 2/20 0.47
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
POLB P06746 1/20 0.46
CDK8 P49336 1/20 0.45
CLK4 Q9HAZ1 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.43
SYK P43405 2/20 0.43
TDP1 Q9NUW8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9683503 0.86 APP (0.62) RAF1MAP2K1APPKDM4EPOLB
SCHEMBL9425740 0.81 CDK8 (0.50) HDAC1HDAC2APPKDM4ECDK8
SCHEMBL9426849 0.80 HDAC1 (0.57) HDAC1HDAC2TDP1
SCHEMBL9426326 0.79 CDK8 (0.68) APPNPC1RAB9ACDK8CLK4
SCHEMBL9426210 0.78 CDK8 (0.47) APPKDM4EALDH1A1NPC1RAB9A
SCHEMBL9425845 0.74 CYP3A4 (0.64) CDK8CLK4
SCHEMBL5606608 0.74 ALOX15 (0.61) HDAC1HDAC2KDM4EALDH1A1NPC1
SCHEMBL12040759 0.72 KMT2A (0.66) KDM4EALDH1A1NPC1RAB9AL3MBTL1
SCHEMBL9425410 0.72 HDAC1 (0.49) HDAC1HDAC2APPKDM4EALDH1A1
SCHEMBL19199578 0.71 HDAC1 (0.49) HDAC1HDAC2APP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5338745-A Alzheimer's disease MITSUI TOATSU CHEMICALS, INCORPORATION (JP) 1994-08-16 US disclosed
EP-0495998-A1 DIHYDROCAFFEIC ACID AMIDE DERIVATIVE AND APPLICATION THEREOF AS MEDICINE MITSUI TOATSU CHEMICALS, Inc. (JP) 1992-07-29 EP disclosed