Acetophenazine

Acetophenazine

SCHEMBL94266

CC(=O)c1ccc2c(c1)N(CCCN1CCN(CCO)CC1)c1ccccc1S2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

DRD2

The experimentally established mechanism targets of Acetophenazine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 known ✓ P14416 7/20 1.00
HRH1 P35367 9/20 1.00
HTR1A P08908 7/20 1.00
SLC6A2 P23975 7/20 1.00
SLC6A4 P31645 7/20 1.00
ADRA1A P35348 7/20 1.00
DRD3 P35462 7/20 1.00
SLC6A3 Q01959 7/20 1.00
KCNH2 Q12809 7/20 1.00
ADRA2B P18089 6/20 1.00
ADRA2C P18825 6/20 1.00
HTR2A P28223 6/20 1.00
HTR2B P41595 6/20 1.00
ADRA2A P08913 6/20 1.00
DRD1 P21728 5/20 1.00
MLNR O43193 2/20 1.00
ESR1 P03372 2/20 1.00
HRH3 Q9Y5N1 2/20 1.00
PTGS2 P35354 1/20 1.00
CYP1A2 P05177 6/20 0.78

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Acetophenazine SCHEMBL29710923 1.00 HRH1 (1.00) HRH1HTR1ADRD2SLC6A2SLC6A4
Acetophenazine SCHEMBL27848793 0.94 HRH1 (0.89) HRH1HTR1ADRD2SLC6A2SLC6A4
Acetophenazine SCHEMBL123792 0.94 HRH1 (0.89) HRH1HTR1ADRD2SLC6A2SLC6A4
Acetophenazine SCHEMBL1155759 0.94 HRH1 (0.89) HRH1HTR1ADRD2SLC6A2SLC6A4
Acetophenazine SCHEMBL123789 0.94 HRH1 (0.89) HRH1HTR1ADRD2SLC6A2SLC6A4
Acetophenazine SCHEMBL20339946 0.94 HRH1 (0.89) HRH1HTR1ADRD2SLC6A2SLC6A4
Acetophenazine SCHEMBL30903895 0.94 HRH1 (0.89) HRH1HTR1ADRD2SLC6A2SLC6A4
SCHEMBL141601 0.92 HTR1A (0.86) HRH1HTR1ADRD2SLC6A2SLC6A4
Acetophenazine SCHEMBL123791 0.92 HRH1 (0.85) HRH1HTR1ADRD2SLC6A2SLC6A4
Carphenazine SCHEMBL1458434 0.89 HRH1 (0.81) HRH1HTR1ADRD2SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 5441 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026106917-A1 EDIBLE TRANSMUCOSAL DRUG DELIVERY METHOD USING AN INTERMEDIATE CAPSULE AS A TEMPORARY VESSEL BioPhysics Pharma, Inc. (US) 2026-05-21 WO claimed
US-12605345-B2 Transdermal drug delivery system BioPhysics Pharma, Inc. (US) 2026-04-21 US claimed
EP-4654963-A1 TREATMENT OF MENTAL ILLNESS VIA ADMINISTRATION OF BUNTANETAP AND ANALOGUES THEREOF Annovis Bio, Inc. (US) 2025-12-03 EP claimed
EP-4618973-A1 METHODS OF SWITCHING NEUROPSYCHIATRIC MEDICATIONS USING ULOTARONT Sumitomo Pharma America, Inc. (US) 2025-09-24 EP claimed
US-20250268841-A1 Trans-Epithelial Membrane Drug Delivery System Masiz, John J. (US) 2025-08-28 US claimed
US-20250191770-A1 COMPUTERIZED DECISION SUPPORT TOOL AND MEDICAL DEVICE FOR RESPIRATORY CONDITION MONITORING AND CARE PFIZER INC. (US) 2025-06-12 US claimed
US-20250179064-A1 BENZOQUINOLONE INHIBITORS OF VMAT2 AUSPEX PHARMACEUTICALS LLC 2025-06-05 US claimed
WO-2025111482-A1 COMPLEXING AGENT SALT FORMULATIONS OF PHARMACEUTICAL COMPOUNDS AT LOW STOICHIOMETRIC RATIOS BEXSON BIOMEDICAL, INC. (US) 2025-05-30 WO claimed
EP-3334725-B1 BROMODOMAIN AND EXTRA TERMINAL (BET) INHIBITOR AND A PROTEIN PHOSPHATASE 2A (PP2A) ACTIVATOR FOR TREATING BET INHIBITOR RESISTANT CANCER DANA FARBER CANCER INST INC (US) 2025-04-23 EP claimed
US-20250120907-A1 Transmucosal Drug Delivery System Masiz, John J. (US) 2025-04-17 US claimed
EP-0367746-A2 Sustained release drug-resin complexes RICHARDSON-VICKS, INC. (US) 1990-05-09 EP claimed
EP-0174342-B1 BRAIN-SPECIFIC ANALOGUES OF CENTRALLY ACTING AMINES UNIVERSITY OF FLORIDA (US) 1989-12-20 EP claimed
EP-0222425-A2 Brain-specific drug delivery UNIVERSITY OF FLORIDA (US) 1987-05-20 EP claimed
EP-0218300-A2 Brain-specific drug delivery UNIVERSITY OF FLORIDA (US) 1987-04-15 EP claimed
EP-0174342-A1 BRAIN-SPECIFIC ANALOGUES OF CENTRALLY ACTING AMINES. UNIV FLORIDA (US) 1986-03-19 EP claimed
WO-1985003937-A1 BRAIN-SPECIFIC ANALOGUES OF CENTRALLY ACTING AMINES UNIVERSITY OF FLORIDA (US) 1985-09-12 WO claimed
EP-0110955-A1 BRAIN-SPECIFIC DRUG DELIVERY. UNIV FLORIDA (US) 1984-06-20 EP claimed
WO-1983003968-A1 BRAIN-SPECIFIC DRUG DELIVERY UNIVERSITY OF FLORIDA (US) 1983-11-24 WO claimed
US-4407800-A TRYPANOCIDES UNIVERSITY OF VIRGINIA ALUMNI PATENTS FOUNDATION (US) 1983-10-04 US claimed
US-4175119-A Composition and method to prevent accidental and intentional overdosage with psychoactive drugs PORTER GARRY L 1979-11-20 US claimed