SCHEMBL9427345

SCHEMBL9427345

C=CCc1ccc(-c2ccc(-c3ncc(O)cn3)cc2F)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 6/20 0.39
GABRB2 P47870 6/20 0.39
CNR2 P34972 3/20 0.39
MEN1 O00255 2/20 0.39
GAA P10253 2/20 0.39
MAPT P10636 2/20 0.39
CNR1 P21554 2/20 0.39
KMT2A Q03164 2/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
ALDH2 P05091 1/20 0.39
AKR1B1 P15121 1/20 0.39
HPGD P15428 1/20 0.39
PPARG P37231 1/20 0.39
PPARD Q03181 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
ALOX5 P09917 3/20 0.38
POLB P06746 1/20 0.38
GABRB1 P18505 1/20 0.38
RXRA P19793 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9449606 0.85 CYP11B1 (0.39) GABRA1GABRB2CNR2MEN1GAA
SCHEMBL8080634 0.83 MEN1 (0.46) GABRA1GABRB2CNR2MEN1GAA
SCHEMBL10525309 0.78 ESR1 (0.45) GABRA1GABRB2CNR2MEN1GAA
SCHEMBL10382097 0.77 MAOB (0.43) MEN1GAAMAPTKMT2AALDH1A1
SCHEMBL9353374 0.76 CYP11B1 (0.38) GABRA1GABRB2CNR2MEN1GAA
SCHEMBL8807255 0.74 RARB (0.59) GABRA1GABRB2CNR2MEN1GAA
SCHEMBL24125046 0.73 KIF11 (0.39) GABRA1GABRB2CNR2MEN1GAA
SCHEMBL10024823 0.73 KIF11 (0.39) GABRA1GABRB2CNR2MEN1GAA
SCHEMBL8992639 0.73 GABRA1 (0.44) GABRA1GABRB2CNR2MEN1GAA
SCHEMBL9245694 0.73 NPC1 (0.65) GABRA1GABRB2CNR2MEN1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5340497-A Ferroelectric liquid crystal MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1994-08-23 US disclosed
EP-0428665-A1 FLUOROPHENYL PYRIMIDINES. MERCK PATENT GMBH (DE) 1991-05-29 EP disclosed
WO-1990015116-A1 FLUOROPHENYL PYRIMIDINES MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1990-12-13 WO disclosed