SCHEMBL9430489

SCHEMBL9430489

COc1cccc2c1c(N1CCOCC1)nc1c(C(N)=NO)ncn12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 4/20 0.39
STK4 Q13043 1/20 0.39
STK3 Q13188 1/20 0.39
TRPM8 Q7Z2W7 2/20 0.38
MTOR P42345 2/20 0.37
PIK3CB P42338 4/20 0.37
PIK3CA P42336 2/20 0.37
POLB P06746 1/20 0.36
USP2 O75604 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
MAPK1 P28482 1/20 0.36
CLK4 Q9HAZ1 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
ALDH1A1 P00352 1/20 0.35
KMT2A Q03164 1/20 0.35
HSD17B10 Q99714 1/20 0.35
MAP2K7 O14733 1/20 0.35
TP53 P04637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9430096 0.89 MTOR (0.43) LRRK2STK4STK3TRPM8MTOR
SCHEMBL9404296 0.81 HTT (0.44) LRRK2PIK3CBPOLBMAPK1SMN1; SMN2
SCHEMBL9404413 0.79 KDM4E (0.41) LRRK2STK4STK3TRPM8MTOR
SCHEMBL9430333 0.73 GABRA1 (0.43) LRRK2STK4STK3TRPM8PIK3CB
SCHEMBL9404393 0.70 ABL1 (0.40) LRRK2STK4STK3POLBMAPK1
SCHEMBL9312142 0.70 POLB (0.40) LRRK2PIK3CBPIK3CAPOLBCYP1A2
SCHEMBL9404501 0.69 RXFP1 (0.53) MTORPIK3CAPOLBUSP2MAPK1
SCHEMBL7320310 0.69 RXFP1 (0.53) MTORPIK3CAPOLBCYP1A2CYP3A4
SCHEMBL9404284 0.68 RXFP1 (0.49) LRRK2MTORPIK3CBPIK3CAPOLB
SCHEMBL7315229 0.64 RXFP1 (0.69) MTORPIK3CAPOLBUSP2MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5371080-A Central nervous system disorders NOVO NORDISK A/S 1994-12-06 US disclosed