SCHEMBL9430795

SCHEMBL9430795

c1cn(Cc2ccc3[nH]cc(CCN4CCC4)c3c2)nn1

nearest known ligand 0.67

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.67
HTR1D P28221 10/20 0.60
HTR1B P28222 10/20 0.60
HTR2A P28223 3/20 0.54
MPO P05164 3/20 0.53
HTR2C P28335 1/20 0.47
BRD4 O60885 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9077110 0.80 HTR1D (0.67) HTR1AHTR1DHTR1BHTR2AMPO
SCHEMBL8784534 0.80 HTR1A (1.00) HTR1AHTR1DHTR1BHTR2AHTR2C
SCHEMBL8506288 0.75 HTR1D (1.00) HTR1AHTR1DHTR1BHTR2AMPO
SCHEMBL734706 0.73 MPO (0.57) HTR1AHTR2AMPO
SCHEMBL26508359 0.72 HTR7 (0.71) HTR1AHTR1DHTR1BHTR2AMPO
SCHEMBL26508398 0.72 MPO (0.94) HTR1AHTR1DHTR1BHTR2AMPO
SCHEMBL26508337 0.72 MPO (0.67) HTR1AHTR1DHTR1BHTR2AMPO
SCHEMBL26508379 0.72 HTR1A (0.75) HTR1AHTR1DHTR1BHTR2AMPO
SCHEMBL26508375 0.72 MPO (0.67) HTR1AHTR1DHTR1BHTR2AMPO
SCHEMBL26508389 0.72 MPO (0.67) HTR1AHTR1DHTR1BHTR2AMPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1994002477-A1 IMIDAZOLE, TRIAZOLE AND TETRAZOLE DERIVATIVES MERCK SHARP & DOHME LIMITED (GB) 1994-02-03 WO disclosed