SCHEMBL9433650

SCHEMBL9433650

C=CC(=O)Cc1cnccc1-c1ccc([N+](=O)[O-])cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.40
ALDH1A1 P00352 4/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C19 P33261 1/20 0.39
TGM2 P21980 1/20 0.39
MAPT P10636 7/20 0.39
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
POLB P06746 1/20 0.38
GYS1 P13807 1/20 0.38
LMNA P02545 1/20 0.38
DAPK3 O43293 1/20 0.37
SLC22A12 Q96S37 1/20 0.36
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
KDM4E B2RXH2 1/20 0.36
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9433405 0.86 PDE4A (0.43) ALDH1A1MEN1KMT2ACYP1A2CYP3A4
SCHEMBL9433930 0.84 GPBAR1 (0.36) ALDH1A1CYP1A2CYP3A4CYP2C19SLC22A12
SCHEMBL9433838 0.83 RPS6KA3 (0.50) KMT2AMAPTRAB9ASLC22A12
SCHEMBL9433512 0.82 SLC22A12 (0.41) ALDH1A1CYP3A4CYP2C19RAB9ASLC22A12
SCHEMBL9434027 0.82 SLC22A12 (0.40) ALDH1A1TGM2MAPTPOLBLMNA
SCHEMBL9433530 0.82 RPS6KA3 (0.35) MAPTSLC22A12
SCHEMBL9433598 0.79 RORC (0.40) L3MBTL1ALDH1A1MEN1KMT2ACYP1A2
SCHEMBL9434303 0.79 SLC22A12 (0.46) ALDH1A1MAPTSLC22A12CYP11B1CYP11B2
SCHEMBL9433809 0.75 GPBAR1 (0.36) ALDH1A1MEN1KMT2AMAPTLMNA
SCHEMBL9434218 0.73 GSTP1 (0.46) ALDH1A1MEN1KMT2AMAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5276150-A Vasodilators, anticoagulants, calcium channel blockers FUJIREBIO INC. (JP) 1994-01-04 US disclosed
EP-0400660-A1 1,4-dihydropyridine derivatives FUJIREBIO INC. (JP) 1990-12-05 EP disclosed