SCHEMBL9433705

SCHEMBL9433705

O=C(C=Cc1cccc2cnccc12)Cc1cccnc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.46
CYP1A1 P04798 2/20 0.46
CYP2D6 P10635 2/20 0.46
CYP1B1 Q16678 2/20 0.46
ALDH1A1 P00352 1/20 0.46
MAPT P10636 1/20 0.46
HPGD P15428 1/20 0.46
NPY1R P25929 1/20 0.46
MAPK1 P28482 1/20 0.46
NPY2R P49146 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
NAPRT Q6XQN6 1/20 0.46
CYP3A4 P08684 2/20 0.42
CYP2C9 P11712 1/20 0.42
TRPV1 Q8NER1 2/20 0.41
IDO1 P14902 3/20 0.40
HDAC8 Q9BY41 2/20 0.40
HDAC6 Q9UBN7 2/20 0.40
HDAC3 O15379 1/20 0.40
HDAC4 P56524 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9434607 0.91 CYP1A2 (0.53) CYP1A2CYP1A1CYP2D6CYP1B1ALDH1A1
SCHEMBL9434718 0.79 NAPRT (0.50) CYP1A2ALDH1A1MAPTHPGDNAPRT
SCHEMBL9434583 0.79 KMT2A (0.49) CYP1A2CYP2D6ALDH1A1MAPTHPGD
SCHEMBL22319877 0.78 CYP1A2 (0.55) CYP1A2CYP1A1CYP2D6CYP1B1ALDH1A1
SCHEMBL9434498 0.78 NAPRT (0.49) CYP1A2CYP1A1CYP2D6CYP1B1ALDH1A1
SCHEMBL9433799 0.78 MAPT (0.61) CYP1A2CYP2D6ALDH1A1MAPTHPGD
SCHEMBL9433617 0.78 HSD11B1 (0.50) CYP1A2ALDH1A1MAPTHPGDNAPRT
SCHEMBL9433573 0.78 NAPRT (0.49) CYP1A2CYP1A1CYP2D6CYP1B1ALDH1A1
SCHEMBL9433920 0.77 TBXAS1 (0.56) CYP1A2CYP1A1CYP2D6CYP1B1MAPT
SCHEMBL3936765 0.77 CDK8 (0.55) CYP1A2CYP1A1CYP2D6CYP1B1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5276150-A Vasodilators, anticoagulants, calcium channel blockers FUJIREBIO INC. (JP) 1994-01-04 US disclosed
EP-0400660-A1 1,4-dihydropyridine derivatives FUJIREBIO INC. (JP) 1990-12-05 EP disclosed