SCHEMBL9433775

SCHEMBL9433775

CSc1ccc([N+](=O)[O-])c(C#N)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VCAM1 P19320 5/20 0.46
MAPT P10636 5/20 0.44
GRIA1 P42261 2/20 0.44
GRIA2 P42262 2/20 0.44
GRIA3 P42263 2/20 0.44
GRIA4 P48058 2/20 0.44
GRM6 O15303 1/20 0.44
CYP1A2 P05177 1/20 0.44
ALOX15 P16050 1/20 0.44
POLB P06746 2/20 0.43
CYP2C9 P11712 1/20 0.43
HPGD P15428 1/20 0.43
APEX1 P27695 1/20 0.43
BLM P54132 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
ALDH1A1 P00352 3/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
KDM4E B2RXH2 1/20 0.39
RECQL P46063 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11335090 0.84 ALDH1A1 (0.41) VCAM1MAPTGRIA1GRIA2GRIA3
SCHEMBL590472 0.80 MAOA (0.61) VCAM1MAPTGRIA1GRIA2GRIA3
SCHEMBL9713754 0.80 MAPT (0.50) VCAM1MAPTGRIA1GRIA2GRIA3
SCHEMBL7281646 0.78 MAOB (0.46) VCAM1MAPTPOLBCYP2C9HPGD
SCHEMBL1343668 0.77 TSHR (0.60) VCAM1MAPTGRIA1GRIA2GRIA3
SCHEMBL8388465 0.77 PDE7A (0.54) VCAM1MAPTGRIA1GRIA2GRIA3
SCHEMBL8390638 0.77 MAOA (0.46) VCAM1MAPTGRIA1GRIA2GRIA3
SCHEMBL592155 0.77 VCAM1 (0.41) VCAM1MAPTGRIA1GRIA2GRIA3
SCHEMBL17870778 0.76 ALDH1A1 (0.55) VCAM1MAPTCYP1A2POLBCYP2C9
SCHEMBL19175487 0.76 DTYMK (0.33) MAPTTDP1ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5350748-A 3-thio or amino substituted-benzo[b]thiophene-2-carboxamides and 3-oxygen, thio, or amino substituted-benzofuran-2-carboxamides as inhibitors of cell adhesion WARNER-LAMBERT COMPANY (US) 1994-09-27 US disclosed