SCHEMBL9433808

SCHEMBL9433808

COC(=O)c1cccnc1C1=C(C)NC(C)=CC1c1ccccc1C#N

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.37
KDM4E B2RXH2 6/20 0.36
HSD17B10 Q99714 2/20 0.36
ALDH1A1 P00352 6/20 0.36
HPGD P15428 3/20 0.36
CRHBP P24387 2/20 0.36
CRHR2 Q13324 2/20 0.36
CNR2 P34972 1/20 0.36
TDP1 Q9NUW8 2/20 0.35
GAA P10253 2/20 0.35
POLB P06746 1/20 0.34
BDKRB1 P46663 1/20 0.34
MAP2K1 Q02750 1/20 0.34
CASP1 P29466 1/20 0.34
CASP7 P55210 1/20 0.34
L3MBTL1 Q9Y468 2/20 0.33
PKM P14618 1/20 0.33
MAPT P10636 1/20 0.33
HTT P42858 1/20 0.33
CYP1A2 P05177 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9433565 0.85 KDM4E (0.38) SMN1; SMN2KDM4EHSD17B10ALDH1A1HPGD
SCHEMBL9434412 0.85 ALDH1A1 (0.40) SMN1; SMN2KDM4EHSD17B10ALDH1A1HPGD
SCHEMBL9433910 0.82 KDM4E (0.44) SMN1; SMN2KDM4EHSD17B10ALDH1A1HPGD
SCHEMBL9434685 0.79 CNR2 (0.39) SMN1; SMN2KDM4EHSD17B10ALDH1A1HPGD
SCHEMBL9434131 0.79 CNR2 (0.34) KDM4EHSD17B10ALDH1A1HPGDCNR2
SCHEMBL9434708 0.78 CNR2 (0.38) SMN1; SMN2KDM4EHSD17B10ALDH1A1HPGD
SCHEMBL9434354 0.77 CNR2 (0.38) KDM4EHSD17B10ALDH1A1HPGDCNR2
SCHEMBL9434469 0.77 KDM4E (0.42) KDM4EHSD17B10ALDH1A1HPGDCNR2
SCHEMBL9433618 0.76 CACNA1B (0.38) KDM4EHSD17B10HPGDCNR2POLB
SCHEMBL9434181 0.76 NPSR1 (0.40) KDM4EHSD17B10ALDH1A1CNR2TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5276150-A Vasodilators, anticoagulants, calcium channel blockers FUJIREBIO INC. (JP) 1994-01-04 US disclosed
EP-0400660-A1 1,4-dihydropyridine derivatives FUJIREBIO INC. (JP) 1990-12-05 EP disclosed