SCHEMBL9434181

SCHEMBL9434181

COC(=O)c1cccnc1C1=C(C)NC(C)=CC1c1cccc(Br)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.40
TSHR P16473 1/20 0.40
POLB P06746 2/20 0.37
RECQL P46063 2/20 0.37
LMNA P02545 2/20 0.37
CNR2 P34972 1/20 0.36
CYP1A2 P05177 2/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
HSD17B10 Q99714 3/20 0.35
KDM4E B2RXH2 2/20 0.35
MAP2K1 Q02750 1/20 0.34
NOTCH1 P46531 1/20 0.34
TDP1 Q9NUW8 2/20 0.34
ALDH1A1 P00352 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
ALOX15 P16050 1/20 0.34
CYP2C19 P33261 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9433618 0.88 CACNA1B (0.38) POLBLMNACNR2MAPTHSD17B10
SCHEMBL9434354 0.84 CNR2 (0.38) POLBCNR2MAPTHSD17B10KDM4E
SCHEMBL9434708 0.83 CNR2 (0.38) NPSR1POLBCNR2GAAMAPT
SCHEMBL9433565 0.82 KDM4E (0.38) POLBCNR2CYP1A2GAAMAPT
SCHEMBL9434685 0.82 CNR2 (0.39) NPSR1TSHRPOLBLMNACNR2
SCHEMBL9433910 0.78 KDM4E (0.44) NPSR1TSHRLMNACNR2CYP1A2
SCHEMBL9434412 0.78 ALDH1A1 (0.40) NPSR1TSHRPOLBLMNACNR2
SCHEMBL9434469 0.78 KDM4E (0.42) NPSR1POLBCNR2HSD17B10KDM4E
SCHEMBL9433808 0.76 SMN1; SMN2 (0.37) POLBCNR2CYP1A2GAAMAPT
SCHEMBL9434784 0.74 CACNA1C (0.41) TSHRPOLBLMNACYP1A2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5276150-A Vasodilators, anticoagulants, calcium channel blockers FUJIREBIO INC. (JP) 1994-01-04 US disclosed
EP-0400660-A1 1,4-dihydropyridine derivatives FUJIREBIO INC. (JP) 1990-12-05 EP disclosed