SCHEMBL9433913

SCHEMBL9433913

COC(=O)C1=C(C)NC(C)=C(c2cccnc2)C1c1cccc(Cl)c1Cl

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 6/20 0.61
KDM4E B2RXH2 6/20 0.61
CYP3A4 P08684 6/20 0.61
CYP1A2 P05177 5/20 0.61
CYP2C19 P33261 5/20 0.61
HSD17B10 Q99714 4/20 0.61
KMT2A Q03164 4/20 0.61
ABCB11 O95342 4/20 0.61
ALDH1A1 P00352 4/20 0.61
HPGD P15428 4/20 0.61
NPSR1 Q6W5P4 4/20 0.61
HIF1A Q16665 3/20 0.61
MEN1 O00255 3/20 0.61
TSHR P16473 3/20 0.61
MAPT P10636 3/20 0.61
CYP2D6 P10635 3/20 0.61
ADORA3 P0DMS8 3/20 0.61
SCN5A Q14524 3/20 0.61
NR1I2 O75469 3/20 0.61
GAA P10253 2/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9434419 0.92 KDM4E (0.49) CYP2C9KDM4ECYP3A4CYP1A2CYP2C19
SCHEMBL9434688 0.89 KDM4E (0.47) CYP2C9KDM4ECYP3A4CYP1A2CYP2C19
SCHEMBL9434014 0.89 KDM4E (0.45) CYP2C9KDM4ECYP3A4CYP1A2CYP2C19
SCHEMBL10432453 0.85 KDM4E (0.49) CYP2C9KDM4ECYP3A4CYP1A2CYP2C19
SCHEMBL9434798 0.84 KMT2A (0.47) CYP2C9KDM4ECYP3A4CYP1A2CYP2C19
SCHEMBL9434605 0.83 NR1I2 (0.52) CYP2C9KDM4ECYP3A4CYP1A2CYP2C19
SCHEMBL9434070 0.83 KDM4E (0.47) CYP2C9KDM4ECYP3A4CYP1A2CYP2C19
SCHEMBL9433574 0.83 KDM4E (0.47) CYP2C9KDM4ECYP3A4CYP1A2CYP2C19
SCHEMBL9434716 0.82 CACNA1F (0.53) KDM4ECYP3A4HSD17B10KMT2AALDH1A1
SCHEMBL29755877 0.82 KDM4E (0.85) CYP2C9KDM4ECYP3A4CYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5276150-A Vasodilators, anticoagulants, calcium channel blockers FUJIREBIO INC. (JP) 1994-01-04 US disclosed
EP-0400660-A1 1,4-dihydropyridine derivatives FUJIREBIO INC. (JP) 1990-12-05 EP disclosed