SCHEMBL9433964

SCHEMBL9433964

COc1cc2c(cc1OC)CN(CCNC(=O)c1ccc([N+](=O)[O-])cc1)CC2

nearest known ligand 0.87

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 3/20 0.71
ABCB1 P08183 2/20 0.71
DRD3 P35462 10/20 0.63
SIGMAR1 Q99720 4/20 0.63
DRD2 P14416 4/20 0.63
DRD4 P21917 8/20 0.60
DRD1 P21728 4/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7167638 0.89 ABCG2 (0.76) ABCG2ABCB1DRD3SIGMAR1DRD2
SCHEMBL9433141 0.85 ABCB1 (0.69) ABCG2ABCB1DRD3SIGMAR1DRD2
SCHEMBL7167644 0.84 ABCG2 (0.59) ABCG2ABCB1DRD3SIGMAR1DRD2
SCHEMBL9433423 0.83 SMN1; SMN2 (0.73) ABCG2ABCB1DRD3DRD2
Bromide SCHEMBL8790411 0.81 ABCB1 (0.62) ABCG2ABCB1
SCHEMBL8789531 0.80 ABCB1 (0.81) ABCG2ABCB1
Hydrochloric Acid SCHEMBL10659282 0.79 ABCB1 (0.80) ABCG2ABCB1
SCHEMBL14721849 0.78 DRD3 (0.79) DRD3SIGMAR1DRD2DRD4DRD1
SCHEMBL10360520 0.78 SIGMAR1 (0.65) ABCG2ABCB1DRD3SIGMAR1DRD2
SCHEMBL8789315 0.78 ALDH1A1 (0.77) ABCG2ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5294621-A Thieno tetrahydropyridines useful as class III antiarrhythmic agents ORTHO PHARMACEUTICAL CORPORATION (US) 1994-03-15 US disclosed