SCHEMBL9433141

SCHEMBL9433141

COc1cc2c(cc1OC)CN(CCNC(=O)c1ccc(N)cc1)CC2

nearest known ligand 0.69

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 2/20 0.69
ABCG2 Q9UNQ0 2/20 0.69
DRD3 P35462 12/20 0.67
SIGMAR1 Q99720 5/20 0.67
DRD2 P14416 4/20 0.67
DRD4 P21917 9/20 0.64
DRD1 P21728 4/20 0.62
TMEM97 Q5BJF2 2/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9433964 0.85 ABCG2 (0.71) ABCB1ABCG2DRD3SIGMAR1DRD2
SCHEMBL7167663 0.84 ABCB1 (0.58) ABCB1ABCG2DRD3SIGMAR1DRD2
SCHEMBL4043245 0.83 SIGMAR1 (0.71) ABCB1ABCG2DRD3SIGMAR1DRD2
SCHEMBL7180280 0.83 SIGMAR1 (0.67) ABCB1ABCG2DRD3SIGMAR1DRD2
SCHEMBL14721849 0.82 DRD3 (0.79) DRD3SIGMAR1DRD2DRD4DRD1
SCHEMBL9433700 0.82 OPRM1 (0.67) ABCB1ABCG2DRD3SIGMAR1DRD2
SCHEMBL4042171 0.81 SIGMAR1 (0.71) ABCB1ABCG2DRD3SIGMAR1DRD2
SCHEMBL8790373 0.81 ABCB1 (0.65) ABCB1ABCG2DRD3SIGMAR1DRD2
SCHEMBL8285666 0.80 SIGMAR1 (1.00) DRD3SIGMAR1DRD2DRD4TMEM97
SCHEMBL9093456 0.79 DRD3 (0.57) ABCB1ABCG2DRD3SIGMAR1DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5294621-A Thieno tetrahydropyridines useful as class III antiarrhythmic agents ORTHO PHARMACEUTICAL CORPORATION (US) 1994-03-15 US disclosed